Caafimaadka, Diyaarinta
Waa kuwee analog "riboksin" Doorto, talooyin iyo dib u eegis
daroogada dhiska - Koox ka mid ah daroogada, hab ugu muhiimsan ee ficil taas oo loogu talagalay kordhaya siin tamarta ee unugyada ee, dardar-korriimadooda iyo kaladuwan, miisaanka oo kordha iyo xawaaraha ee geeddi socodka dheefshiidka. Mid ka mid ah wakiilo ka socda kooxda this daroogada waa "Riboxinum".
sifooyinka pharmacological daroogada
Diyaarinta "Riboxinum" ka dhigan tahay wax soo saarka, daawooyinka ah dhiska, saamaynta ugu weyn ee kaas oo la faray in la kordhiyo iska caabin ah unugyada xaaladaha hypoxia. Sida maamaan ah triphosphate adenosine, "Riboxinum" oo ku lug leh nidaamka cholesterol of glucose gudahood cell iyo, sidaas awgeed, formation of triphosphate adenosine, taas oo substrate ugu weyn ee tamarta cell. In view of this saamayn ah "Riboxinum" fulyo saamayn anti-hypoxic eego hoos content ee ATP.
saamayn dhiska "riboksin" muujiyey by hababka dheefshiidka kordhay lug acid pyruvic iyo dardargelinta ee dehydrogenase xanthine. Sababo la xiriira saamaynta kuwan "Riboksin" leedahay saamayn togan ku saabsan koorsada of saamaynta dheefshiidka unugyada gudahood, kor u qaadida sahayda tamarta ay hawlgal caadi ah.
Markii loo feydo myocardium ah "Riboxinum" optimizes myocardiocytes, qayb dheeraad ah oo buuxda ay nasashada (kordhaya phosphorylation ee bonds actin-myosin ah) iyo sidoo kale shidaa habka regenerative ee myocardium ah.
In la eego geedi socodka pharmacokinetic "Riboksin" si fiican u quudiyey galay wareegga systemic durba Lumen ee mareenka caloosha iyo mindhicirka. Waayo, jidadka parenteral maamulka (i.v.) "Riboxinum" ku filan si degdeg ah loo qaybiyey unugyo marinkii marxaladaha xiga ee unugyada dheefshiidka beerka, halkaas oo in ay ka baxayaan buuxa. Digo ee metabolites unmetabolized oo u taagoo daroogada waxay dhacdaa inta badan kaadida, iyo qayb yar oo ka qayib saxarada iyo bile.
Tilmaamayaasha
Drug "Riboksin" ayaa tilmaamay in daaweynta cudurada wadnaha, oo ay ku jiraan kuwa lagu daaweyn jiray wadamada post-Wadnaxanuun. daroogada waxay leedahay saamayn ku daweyn wanaagsan ee daaweynta ee dalalka of laxanka iyo tabinta rabshooyin, badinta diyaarinta of wadnaha glycosides, daaweynta cilladaha morphological ee muruqa wadnaha, taasoo keentay in asalka ah ee kor u load jirka, ama ka dib cudurada faafa iyo bararka.
"Riboxinum" muujiyay therapy cudurada nidaamka hepatobiliary, waayo, ka hortaga cudurada nidaamka dhiigga ee diyaarinta qaadasho sare ee shucaaca ionizing. In dhaqanka indhaha, isticmaalka "riboksin" roon at glaucoma-xagal furan.
"Riboksin": tilmaamaha loo isticmaalo, analogs
Marka la isticmaalayo qaab kiniin oo ah daroogada waa inay raacaan talooyinka. Waayo, dadka waaweyn, qiyaasta maalin kasta ee daawada u dhaxayn kartaa 0.6 2.4 grams. Sida caadiga ah, qiyaasta waxaa si gaar ah u Hagaajinay, iyo qiyaasta maalin kasta waxaa loo qaybiyaa dhowr jeer maalintii oo dhan. kiniin la magacaabo waa inay ahaadaan qiyaasta ugu yar, iyo kaliya hadii qiyaasta ugu yar waxaa caadi ahaan loo dulqaatay by bukaanka, ka dib markii 2-3 maalmood kicin. Duration ee therapy waa in laga bilaabo 1 illaa 3 bilood.
In maamulka parenteral, xal 2% "Riboxinum" a qasi 250 mL ee biyaha cusbada chloride sodium ama glucose. galiyey waxaa lagu fuliyaa si tartiib ah heer ah 40-60 dhibcood halkii daqiiqo.
analogs dheeraad ah oo la mid ah Qiyaasta waa in la ogaadaa, "Inosine" iyo "Ribozin", taas oo hoos laga wada hadli doono.
Sababo in daroogada
Sababo si ay u bixiyaan dareen korodhka in mid ama ka badan qaybaha daroogada, turqo iyo heerarka sare ee acid uric ee plasma dhiigga. Iyada oo taxaddar dheeraad ah waa in la qoray "Riboksin" iyo analoogga "riboksin" bukaanka "Inosine" la failure of function excretory kelyaha.
waxyeellooyin
Caadi ahaan, daawada waxaa si fiican loo dulqaatay. Ka mid ah kuwa ku arkay dareenka sii kordhaya in ay daroogada oo laga dheehan karo ka maqaarka xajiinta. On qayb ka mid ah nidaamka wadnaha iyo waxay keeni kartaa wadno, kordhay cadaadiska dhiigga, daciifnimo.
Haddii ay dhacdo in bukaanka qaata 'Riboksin "arkay dhibaatooyinka kor ku xusan, waa in aad Takhtarkaaga la tasho iyo joojin qaadashada daawada.
tilmaamaha gaarka ah ee qaata
Tan iyo markii ay "Riboxinum" iyo metabolites ay raaca inta badan by kelyaha, ma ku haboon yahay isticmaalka daroogada ay goobjoog ka ahaayeen renal failure. Isticmaalka daroogada this xaq ku noqon karaa oo kaliya in kiiska halkaas oo faa'iidada laga filayo daroogada badan halista ka iman karta ay isticmaalka weyn. Hoggaansamaan xeerarka la mid ah in magacaabidda daroogada si uu haweenka uurka leh iyo kuwa nuujinaya.
Marka la eego saamaynta "riboksin" on heerka acid uric ee plasma dhiigga inta lagu jiro daaweynta waxaa lagu talinayaa in ay la socodka joogtada ah si looga hortago dhacdo ee hyperuricemia.
Sunta iyo badinta daroogada
In case of qaata qaadasho sare ee medicament qaadeen tallaabooyin guud golleeyahay in lagu yareeyo daroogada galaya dhiigga. In case of calaamadaha lagu sumoobo - therapy astaamaha. Marka dareen diidmo oo xasaasiyadeed, therapy sadha waa wax ku ool ah.
"Riboksin": dhigooda
Si aad u taariikhda, suuqa dawooyinka ma jiro mid ka mid analoogga "riboksin" with hab dhiska garoomada. Xaaladdan oo kale, waxaa jira labada analogs ku jirto qayb kale oo firfircoon, iyo sidoo kale micne ah dhamaystiran oo daroogada, waxay leeyihiin in la mid ah qayb firfircoon ay ka kooban.
"Inosine" Waxaa laga yaabaa in isku iyo analog buuxa "Riboxinum" maamulka muruqyada dhexdooda. At ay asaasiga ah, daroogada waa bedel buuxa for "riboksin" oo dhan tilmaamo iyo sababo ay. micne tixgeliyo kale daroogada - "Ribonozin". diyaarinta Tani waxay sidoo kale waxaa ku jira qayb firfircoon, daawo la mid ah "Riboksin" ee ay ka kooban. Analoogga ee carruurta ee sharoobada - daroogada sida "Mildronat". Waxa uu sidoo kale awood u leh inay siiyaan homeostasis tamarta ee dhowaad dhammaan unugyada jidhka ku.
Haddii aan ka fiirsan kooxda daroogada dhiska non-steroidal, waxaan kala saari karaa analogs sida kiniinno "Riboxinum" sida "Methyluracil" iyo orotate potassium. Daawooyinkan, inkasta oo ka tirsan kooxaha pharmacological kala duwan, si kastaba ha ahaatee, waxay awoodaan inay tijaabiso saamayn dhiska. Guud ahaan, saamaynta this waxaa sabab u ah kicinta ah ee geedi socodka dheefshiidka in dhammaan unugyada iyo unugyada jirka.
Barbar Dhigo daroogada "Riboksin" dhigooda cusub Qarni, waxaan la soco in ay leeyihiin oolnimada sare iyo saamaynta-ku-daweyn. Wakiil ka mid istaahila in kooxdan waa "Citoflavin". analoogga "riboksin" Intaa waxaa dheer Tani waxay saamayn cytoprotective iyo antioxidant oo uu leeyahay saamayn dhiirrigelin xoog on neurons maskaxda.
gunaanad
daroogada dhiska - daroogada koox ballaaran oo qaab-dhismeedka kiimikada kala duwan. Iyada oo ku xidhan ujeedada taas oo aad qorsheyneysid inaad ku isticmaasho, waxaad dooran kartaa "Riboksin" analogues daroogada, ama bixiso kooxda steroid fiiro dheeraad ah. Ogsoonow in aan la talinayaa codsiga madax banaan daawooyinkan. takhasus gaar ah u qalma oo kaliya ayaa kaa caawin kara in doorashada ee daroogada.
Similar articles
Trending Now