Caafimaadka, Diyaarinta
"Luminal": tilmaamaha isticmaalka dhashay
Waa maxay daawada "Luminal"? Tilmaamaha iyo tilmaamo ah daroogada this la hoos ku hadli doonaa. Waxaan sidoo kale qeexi guryaha pharmacological sida daroogada, saamaynta dhinaca iyo sababo.
Halabuurka The daroogada iyo qaab
Taasi waxaa ku jira daroogada ah "Luminal"? Tilmaamaha loogu isticmaalo ayaa sheegay in in ka kooban of dejinta waxaa ka mid ah qayb firfircoon sida phenobarbital. hab sidoo kale loo arkaa ka mid ah kuwa soo socda qaybaha dheeraad ah: istaarijka baradho, gelatin, Rusheyn kartaa oo ku milmahayn calcium.
Diyaarinta "Luminal", tilmaamo ah kuwaas oo la oran soo bandhigay, waa suuq foomka budada ah loogu talagalay xal la isku duro. Sidoo kale qalab laga iibsan karaa qaab kiniin oo ah 100 mg, kaas oo lagu buuxiyey oo ku yaal dusha cell iyo Baakadaha warqad sameeyey, siday u kala horreeyaan.
Saamaynta daweynta ee daroogada
Waa maxay daawada sida "Luminal"? Tilmaamaha loogu isticmaalo doodaysaa in daawaynta this ayaa ku dejinaysaa, hypnotic iyo saamaynta anticonvulsant.
Viewed medicament awood dadkaas tallaabo suppressive (non-xulashada) ee habdhiska aadanaha, iyo sidoo kale la xakameeyo deegaanka qaarkood (sida caadiga ah dareen) kiliyaha yareeyo hawl socon karto, horumarinta Lulmo iyo hurdo.
Drug "Luminal" edbinta ku saabsan codsiga ah ee ku taal dalka xidhmooyin warqada waa barbiturate aad u xoog badan. guryaha ku dejinaysaa-hypnotic Its waa ay sabab u tahay Iscelin of hawsha unugyada, oo aad dhaqaajiso formation reticular ah oo ka mid ah nuclei of thalamus, jiridda maskaxda ah, oon ku joogsada dhexgalka yidhi dhismayaasha la kiliyaha cerebral.
Features daroogada
Waa maxay daawada cajiib ah "Luminal"? Tilmaamaha loogu isticmaalo (dhallaanka waa hab qoray marar aad u badan) waxa uu dhigayaa in hurdada ay keento barbiturate this, marka la barbar dhigo kula biyaha cusbada ayaa qaab ka duwan. Sida caadiga ah, horumarinta saamaynta hypnotic ka dib codsanaya dawadan loogu talagalay 35-65 daqiiqo muddo 6-9 saacadood.
Waxaan ma dhihi karo in daawaynta hoos tixgelin bandhigaa kaga hadlay guryaha anticonvulsant. Waxaa sababa saameynta ay daroogada meelaha qaar ka mid ah habka dareemayaasha jirka. Marka la isticmaalayo daroogada this ee bukaanka hoos excitability neuronal aaga epileptogenic taasoo ka hortagaysa soo bixitaanka iyo faafinta ee la karsado. Sidoo kale asalka ah "Luminal" ayaa sheegay in ka xanibeen siideeyn ee hirka sare ee neurons, korodhka marinkii dareenka korontada ee gobolka motor of kiliyaha cerebral ah.
Intaa waxaa dheer, waayo, daroogada la siiyey waxaa lagu gartaa saamayn xanuunka yar iyo antigiperbilirubinemichesky. Sidoo kale ayaan meesha ka saarin xoojinta celintan jirka ee ku meersan waxa daran.
qaadashada Small "luminal" leeyihiin saamayn ku dejinaaya, iyo xarumaha sare medulla neefta -ugnetayut iyo t. D.
Tilmaamo ogeed
haddii daroogada la nuugo, "Luminal"? Tilmaamaha loogu isticmaalo ayaa sheegay in jirka gudihiisa waxaa Oo Qaliin nuugista a gaabis ah oo dhamaystiran. bioavailability ee wakiilka uu ka yahay ilaa 80%, iyo bond si borotiinada plasma - oo ku saabsan 30%.
Walaxda firfircoon ee daroogada guskiisa caanaha hooyada, iyo sidoo kale mandheerta. Intaas waxaa sii dheer, waxaa loo qaybin karaa unugyada uurjiifka.
Digo "luminal" dhacdaa via kelyaha qaab beddelin ama qaab metabolites. Waayo, phenobarbital lagu gartaa raasamaal arrin wayn. Xanuunka of kelyaha sababa dheereyn tallaabo.
Drug "Luminal": muujinaya in loo isticmaalo
Waxaa loo tixgeliyaa daroogada la qoray dadka waaweyn oo keliya ma aha, laakiin carruurta iyo dhallaanka. Sida caadiga ah, waxaa loo isticmaalaa:
- hyperbilirubinemia;
- qalalka,
- teetanada (waayo, therapy Waxuu curiyaha);
- daaweynta qalal convulsive ba'an.
Waxaan ma dhihi karo in qalab this ahaan loogu talo galay daawaynta la isu geeyey sida daroogada ah ku dejinaysaa si loo baabi'iyo welwelka, cabsida iyo walwalka.
Oo mamnuucday isticmaalka
Haddaba aad u ogaato waxa xaaladda bukaanka waxaa qoray daawo ah "Luminal". Tilmaamayaasha ay u isticmaalaan daroogada this lagu kor ku xusan. Iyadoo la tixgelinayo sababo ah, ka dibna ay fuliyaan sida:
- dareen sare si ay daroogada,
- beerka daran iyo kelida oo dhaawac gaaro;
- noocyo kala duwan oo porfyri;
- nuujinta iyo uurka.
Medicament "Luminal": tilmaamaha loo isticmaalo carruurta iyo dadka waaweyn
Isticmaalka daroogada this waa in si adag loo tilmaamay. Its isticmaalo waxay u baahan tahay doorashada ee mudada shakhsi daaweynta, qiyaasta, iyo mudada taas oo ku xiran ma aha oo kaliya on nooca socodka cudurka, laakiin sidoo kale on da'da bukaanka iyo sifooyinka kale.
Sida laga soo xigtay tilmaamaha, qalabka celcelis ahaan qiyaasta warbixineed hal ee dadka waaweyn waa 10-200 mg. Qaado kaniiniga sida waa in ay ahaataa 1-3 jeer maalintii.
Sida loogu talagalay carruurta dhasha, iyaga qaadashada daawada waxaa loo xisaabiyaa ku salaysan miisaanka jidhka (miisaanka 1-10 mg / kg jirka saddex jeer maalintii).
Haddii loo isticmaalaa in lagu foomka cudurada of galiyey daroogada daweeyo, qiyaasta dadka waaweyn waa 100-1400 mg (faleebo gale), ama 10-200 mg (for duridda).
Xisaabinta qiyaasta mawduuca daawada carruurta waxaa sidoo kale lagu sameeyaa ku salaysan miisaanka ilmaha.
Sida laga soo xigtay khubaro ah, ka dib markii maamulka xididka, "luminal" ay saamayn ugu badnaan la gaaro 35 daqiiqo gudahood.
waxyeellooyin
Ma saamayn xun ku daroogada aadanaha jirka "Luminal"? Tilmaamaha loogu isticmaalo (xasaasiyadda ka dhigan tahay in aan lagu tilmaamay) doodaysaa in daaweyn jiray xogta daawada bukaanka waxaa laga yaabaa in la horumariyo noocyo kala duwan oo waxyeelo wada khuseeya xubnaha muhiimka ah iyo nidaamka. calaamadaha Dacdarrada daciifnimo, daal, hurdo la'aan, niyad-jabka iyo ataxia. Waxa kale oo suuragal horumarinta Torombositobiiniya, Agranulocytosis, dareen diidmo oo xasaasiyadeed iyo cudura shiid calcium.
xaaladood oo badinta
Iyada oo ah qiyaasta xad dhaafka ah ee bukaanka "TMB" aad inta badan madax xanuun, nystagmus, dawakhaad, ataxia, dhibaato neefsashada, feejignaan xumo, daciifnimo, dhantaalan hadalka, hurdo, isbeddel ah ee heerkulka jidhka, kacsiga, cadaadiska dhiigga iyo fashilaad kale. Xaaladaha aad u adag, waxaa ka mid ah: bradycardia ama tachycardia, barar sambabada, wareer, garaaca, kooma, pneumonia iyo wixii la mid ah.
Si aad u baabi'iyo calaamadahan waa lavage qoray gastric iyo sidoo kale daaweynta naanin ah.
isdhexgalka daroogada
Codsiga of wakiilka loo arkaa in isku darka daawooyinka laga diiqadoodo HC, methylphenidate ama inhibitor MAO kordhiyaa-fiirsashada ee ay qayb firfircoon ka kooban ee plasma ah, taas oo horseedaysa in ay kor u saamayn sun iyo Iscelin of NA ah.
isku darka ah "Luminal" la corticosteroids, chloramphenicol, corticotropin, dacarbazine, Cyclosporine, glycosides digitalis, quinidine, metronidazole, murugada tricyclic, carbamazepine, anti-qabashada, tirsan group succinimides, doxycycline, xinjirowga lidka ku ah, chlorpromazine, fenoprofenom, vitamin D iyo phenylbutazone yarayn karaa muddada tallaabo iyo xoojinta daroogada, kuwaas oo kor-shiid, iyo sidoo kale culayska saaran beerka.
daaweynta oo raacsan ka acetazolamide taraysaa in ay horumarinta rickets iyo osteomalacia. Valproic acid kor u fiirsashada phenobarbital ee dhiigga, taasoo keenta suuxin a fahmayaan iyo feejignaan xumo.
Isticmaalka "luminal" si wadajir ah ula nimodipine, "Verapamil" iyo felodipine yaraynaysaa ay fiirsashada ee dhiigga.
isku dhafan ee medicament la maprotiline wanaajisaa saamaynta ay inhibitory on NA ah, waxay yaraysaa saamaynta barbiturates anticonvulsant oo marinka convulsive.
Walaxda Firfircoon "luminal" paracetamol waxay yareyn kartaa tayada iyo kor u qaado horumarka of hepatotoxicity. Marka lagu daro folic acid yaraynaysaa oolnimada of phenobarbital.
Pyridoxine hoos u fiirsashada dhiigga phenobarbital, iyo primidone, felbamate iyo, taas bedelkeeda, waxaa kor loogu qaado.
Analogs oo ka mid ah daroogada iyo qiimaha
Daawada aasaasiga ah waxaa loo arkaa analogues hab sida "Barbinal" iyo "Dormiral".
kiniiniyada Kharashka "Luminal" (100 mg, 10 kumbiyuutarada.) Of 1100 rubles iyo wixii ka sareeya.
macluumaad gaar ah
soo dhaweynta wadajira "luminal" ka ethanol iyo ethanol-hab si weyn kor loogu qaado karaan saamaynta inhibitory daroogada on habka dareemayaasha jirka bukaanka. Sidaa darteed, cabitaanka khamriga iyo tinctures kale, daawooyinka ku saabsan khamriga inta lagu guda jiro daawaynta wakiilada kuwan yihiin.
Reviews
dib u eegista Inta badan diyaarinta this tago waalidka caruurta yar yar. Waxay ku doodayaan in daroogada "Luminal" Dagaalka wanaagsan oo cudurro sida qalalka iyo xaaladaha convulsive. Waxaa sidoo kale inta badan daawooyinka waxaa loo isticmaalaa oo qayb ka ah therapy isku dhafan, dhamaystir u xanuun joojiyaha uu.
bukaan badan ayaa sheegaya in tayada sare ee daroogada "Luminal". Si kastaba ha ahaatee, waxay si deg deg ah ku xusan in la helo dul lacagta waa in si adag raacdo qiyaasta iyo isku dhafan oo daroogo kale.
Mararka qaarkood loo arkaa daawo loo isticmaalo daweynta dadka qaba dystonia vascular, kaas oo la Ulasocto joog- weerarada argagaxa. Daaweynta qalab this ka caawisaa in ay caadi xaaladda bukaanka, gaar ahaan haddii ay ahayd daawo dheeraad ah, weynaadaa xididdada dhiigga iyo yareeyaa dubaaxin.
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