Caafimaadka, Diyaarinta
"Stamlo": dib u eegista, analogs. Tilmaamaha loogu isticmaalo "Stamlo"
Si aad u cadaadiska dhiigga hoose, dhakhaatiirta inta badan ay isticmaalaan daawooyinka oo ku salaysan amlodipine. Mid ka mid ah hab oo kale waa daroogada ah "Stamlo".
description
daroogada Tan waxaa loo sameeyey by shirkad Hindi ah, "Dr. Reddy ee Laboratories Ltd.".
Daawo "Stamlo" muujinaysaa saamayn dose-ku-tiirsane ah oo daba dheeraata daweynta.
Sida dihydropyridine derivative qayb amlodipine jilitaanka ah loola jeedaa jiilka labaad Ca 2+ ku Doodeen, taas oo ay xirto ee channels, udhigo calcium transmissive.
foomka qiyaasta
hab la heli karo in labo qaadashada: 0.005 iyo 0.010 g of qayb walax firfircoon.
dose Hoose ee medicament "Stamlo" edbinta ku tilmaamay sida kiniinno wareega leh dusha cad ama si xooga cad, taas oo ah guri, geesaha uu leeyahay qaab chamfered. Ujeedada calaamadeeysid daroogada waxaa ku jira isla extrusion diyaarad «ah R 177", oo dhinaca kale ah - codsatay in ay halis kala.
Qiyaas badan ee daawada "Stamlo" qeexayaa aan la taaban karin sida kiniin ah gadood la dusha cad ama ku dhowaad caddaan biconvex. Ujeedada calaamadeeysid daroogada ka mid ah diyaarada waxaa Tuujiya «R», oo dhinaca kale ah - waxaa laga codsadaa, tireedyada tixraaca "178". unugyada qiyaasta adag ayaa laga heli karaa baakad fin of 14 xabbadood ee baakad ay ku jiraan xirmo laba doonistiisu ahayd.
qaybaha daroogada
Walaxda firfircoon ee daroogada waa cusbo ah nooca besylate amlodipine, qadarkuu of 6,42 mg iyo 12,838 oo u dhiganta 0,005 oo 0,010 g of amlodipine saafi ah.
In qaabka kiniinka "Stamlo" ogaan karaa qaybaha aan firfircoonayn, kuwaas oo wakiil ka qayb of mikrokristallin nooca cellulose, sodium glycolate noqde, aerosil fuuq, milmahayn magnesium.
hab of action
Taagoo ku xidhaan in channels qufulka nooca outgrowths amlodipine receptor dihydropyridine lays gaabiska ah ee atammada kalsiyamku ay leeyihiin lakabka labaad oo bixiya antihypertensives iyo dhaqdhaqaaqa antianginal.
Tilmaamaha loogu isticmaalo "Stamlo" waxaa lagu tilmaamay sida dawo, taas oo qabata transmembrane guurka hoos Ca 2+ udhigo unugyada muruqa siman derbiga vascular.
Marka hawlaha antianginal furaaya weelashii halbowlaha wadnaha waaweyn iyo kuwo yaryar iyo nooca durugsan. In joogitaanka xanuun laabta ah hoos u astaamaha gobolada ischaemic muruqyada wadnaha.
daroogada waxay bixisaa saamayn daciif natriuretic, Iscelin of xulkii dhiig xinjirowga unugyada, kordhiyay heerka sifeynta glomerular.
Expansion ee arterioles fog sababa hoos u dhac ku caabin guud ee sariirta dhuumaha ugu sarreeya, loader hoos on nudaha cajiib ah myocardial, yareynta qadarka oksijiin kelli looga baahan yahay wadnaha.
Reception ka dhigan tahay bukaanka qaba nephropathy diabetic ma Microalbuminuria inta badan sameysa.
tallaabo ee daroogada uusan u beddelmin oo heerka shiid iyo la egyahay ee dhiigga.
hawl-daweynta dhacdaa dhowr saacadood ka dib loo dhawray hal maalin.
Maxaa loo isticmaalaa
Kiniinka caawin xanuun laabta dawayn iyo dhaqdhaqaaqa jirka lama filaan ah.
Tilmaamaha loogu isticmaalo "Stamlo" talinaysaa qaadashada for cadaadis dhiig oo sareeya. Waa in la keli ahaan ama isku darka daawada kale antihypertensive isticmaali karaa.
Sida loo qaato
Kiniiniga "Stamlo M" diiwaanka ku talinaysaa in lagu daweeyo halbowlaha dose bilaabo xaalad iyo xabad xanuun hypertensive ee 0,005 g of cabitaan in 1 jeer maalintii. Caddadka taageerada of amlodipine at cadaadis kacsantahay waa 0,005 garaam maalin kasta. ugu badnaan ogol yahay qiyaasta maalin walba ah ee lacagta waa in aanay ka badan 0,010 g
Lama filaan ah oo angina inta lagu guda jiro jimicsi dose daawo ee ka soo 0,005 in 0,010 g maalintii.
Inta ay sixida medicament "Stamlo M" waxa aan sameeyaa haddii la isku daro la diuretics thiazide, angiotensin diinta retarders enzyme, daawooyinka amooniyam adrenoblokatornymi beta iyo saamaynta dheer iyo nitroglycerin sublingual.
Marka hawlaha hypotensive bukaanka da'doodu tahay, la koritaanka yar, la mass muruqa hooseeyo, cillad ah ee beerka waxaa loo isticmaalaa in marka ugu horeeysa ee medicament 0,0025 Waayo, bukaanka noocan oo kale ah, qiyaasta waxa lagu tilmaamayaa loogu daweeyo antianginal at 0.005 g
Haddii ay jirto failure a of kelyaha, ka dibna la qabsato xaddiga amlodipine muhiim ma aha.
Features ee daaweynta
By daroogada "Stamlo" edbinta ku saabsan wararka ku saabsan suurtagalnimada of adeegsigeeda bukaan badan oo monotherapy. Haddii ay jirto la'aanta hawlaha antihypertensive, waxaa lagu darayaa diyaarinta inhibitors enzyme angiotensin-beddelaya, diuretics xubno thiazide, daawooyinka adrenoblokatornye Alfa iyo beta.
Inta lagu guda jiray daawada waxay u baahan tahay la socodka miisaanka jidhka aadanaha iyo qaadashada sodium, talooyinka cuntada waa in la raaco.
Oo looxyadu waxay ka mid noqon kara monotherapy, ay weheliso daroogada hawl antianginal ee bukaanada madax adkaadeen, si ay saamaynta qaadashada daweynta amooniyam iyo walxaha beta adrenoblokatornyh.
Si looga hortago dhiig bax, xanuun iyo juqda unugyada ee ciridka, ilkaha prophylaxis u baahan yahay booqashooyin joogto ah oo wareegsan ilkaha.
Maadadaha xannibi lays gaabiska ah ee atammada kalsiyamku dhex channels ah ma keenaan jawaab jirka ee la kansalay ee medicament ah, laakiin-daaweynta aan waa in si tartiib tartiib ah loo yareeyo qiyaasta.
content ee siifilisku potassium, glucose, kolestaroolka, taagoo triglyceride, uric acid iyo kariyaatiniin ee dhiig ma kala duwan yihiin sarkhaansan yihiin kiniiniyada "Stamlo".
In marxaladaha hore ee daaweynta, bukaanka waxaa laga yaabaa in hurdo ama dawakh, taas oo u baahan taxadir inta lagu guda jiro wadista gaadiidka.
Yaa waa in aan qaato
Tilmaamaha loogu isticmaalo "Stamlo" qasab ku jira liiska sababo, kaas oo bukaanka aan qoray kaniiniga. Kuwaas waxaa ka mid ah:
- hypotension halbowlaha in u daran marka index cadaadis systolic ka hooseeyay 90 mm Hg;
- kollapsicheskoe iyo gobolka shoog cardiogenic;
- feedho xanuun aan daganayn, marka lagu daro muuqaalka lama filaan ah;
- xilliga dhalmada iyo naas-nuujinta;
- dareen xad-dhaaf ah si ay maaddooyinka oo ka mid ah xeryahooda daawo iyo dihydropyridine.
- Ha isticmaalin qalab ilaa 18 sano jir, sida ay aan la xaqiijiyay waxqabad ammaan ah.
U baahan tahay taxadar in isticmaalka bukaanka qaba failure nooca dekompensatsionnaya muruqa ah chronic wadnaha, quruxsan jilicsan ama dhexdhexaad ah oo ah dhiig-karka, aortic iyo mitral foomka vasoconstriction, myocardial infarction cajiib ah, sonkorta xad-dhaaf ah oo ba'an, xadgudub ah ee beerka iyo shiid dufanka.
dhibaato
on codsiga ee buuga "Stamlo" sheegaye oo dhan cawaaqib xun, dhacdo taas oo suurto gal ah ka dib markii qaadashada daawada.
At nidaamka wadnaha iyo xididdada ayaa wax ku ool ah ee amlodipine la dhalashada of garaaca wadnaha ah, neefta oo ku qabata, decompression cad, syncope, reaction vaskulitis, barar habka lugaha hoose iyo hubka.
On habka nidaamka dawada habdhiska neefsashada iyo hawl la dhacdo xanuun madaxa, daal, isbedellada niyadda, suuxid, neefta oo ku qabata, murugada, qufac ama rhinitt.
Laga soo bilaabo daawada matag karo, mantag, calool xanuun, horumarinta ganaca, gastritis iyo cagaarshow, afka oo qalala, peristalsis jabay, kordhin fiirsashada of falgalka cagaarshowga.
Isbedelada nidaamka Fistula, muujiyey by rabitaanka soo noqnoqda ama xanuun peeing, xanuunada dheecaanka, Nocturia, hoos u awoodba.
Falcelinta maqaarka la xiriira xeroderma timaha, purpura, astaantii oo ka mid ah xasaasiyad epithelium, pruritus, finan, anjioedema.
On habka amlodipine muruqyada si xun u saameyn muuqaalka kore ee arthralgia, arthritis, dhabar xanuunka iyo tabar-dari muruq.
xubnaha dareenka kara dhibaatooyin xagga horumarinta aragga oo labalaabma, caabuq conjunctiva ah, xanuunada indhaha iyo dareenka aragtida dhadhanka, dhaguhu madaxa, hoy indhaha, qallayl oo ka mid ah wilka iyo xuub-axaleedka.
Sidee si ay ula falgalaan daawooyin
Lifaaqsan medicament ah "Stamlo" tilmaamaha isticmaalka kiniinka aan lagula talinayaa in lagu biiriyo walxaha in la xakameeyo qayilo ee microsomal. Under saameynta ay, waxay kordhisaa heerka plasma of amlodipine, kordheen tirada geedi socodka la rabin. Isku dhafan oo inductors oo dardar-falgalka microsomal cagaarshowga, saamayn ka soo horjeeda.
dhaqdhaqaaqa Antihypertensive waxaa wiiqday sarkhaansan yihiin daroogada anti-bararka magnyl. sodium indomethacin raagay iyo Avv prostaglandin laga xannibo in kelyaha, iyo Alfa-agonister sidoo kale estrogen hoos Digo ee udhigo Na +, waa saamayn sympathomimetic.
Warfarin, digoxin, cimetidine iyo pharmacokinetic qiyamka ma beddeli dabeecadaha Alwaaxdii.
Antianginal iyo ficil hypotensive la xoojiyo karaa thiazide, "loop" diuretics, hab beta-adrenoblokatornymi, verapamil, angiotensin diinta inhibitors enzyme, iyo Nitrate.
Walxaha ka kooban Ca 2+ udhigo, blokatorny hoos saamayn on channels calcium.
Astaanta of saamaynta neurotoxic daawooyinka lithium maqalka amlodipine, taas oo ah waxa lagu gartaa lallabo, shuban, matag, gariirka, ataxia, tinnitus.
Amiodarone, Alfa-blockers, quinidine, walxaha neuroleptic waallida dajiya daroogada nooca korodhka dhaqdhaqaaqa hypotensive.
isticmaalka xad-dhaafka ah
Iyada oo ah qiyaasta xad dhaafka ah ee hagaha daroogada "Stamlo" qeexayaa isbedel, lagu gartaa hoos u cad in cadaadis, foosha noqnoqda ee wadnaha, vasodilation durugsan xad-dhaaf ah.
hawlaha ayaa sidoo kale loo arkaa in ay ka saarto lavage la xiriira daroogada xad gastric, magacaabidda sorbents. Waxaa muhiim ah in la soo celiyo dhaqdhaqaaqa ee weelashii sambabada, wadnaha iyo dhiig, si ay ula socdaan waxqabadkooda. Waa in lagu hayo gobolka wanaagsan oo addimada, si loo xakameeyo mugga of kaadida.
Kuwa caburka waxaa loo isticmaalaa caadi ah ee midab vascular. Si aad u baabi'iyo saamaynta embriyaha qufulka intravenously calcium waxaa loo isticmaalaa sida gluconate ah.
daawooyinka la mid ah
Waayo, daroogada analogues "Stamlo" ayaa sidoo kale lagu heli karaa laba qaadashada: 0.005 iyo 0.010 g of amlodipine. Halabuurka The oo tayo leh oo ka mid ah waxyaabaha aan firfircooneyn ee kiniinka ka saarayaasha kala duwan wax yar kala duwanaan karaan, uusan saamayn ku lahayn bioavailability ah.
Drug "Amlodipine" soo saaray "ALSI Pharma" CJSC. Waxaa loo tixgeliyaa mid ka mid ah analogues Indian raqiis ah daroogada. Waxay leedahay hawl antianginal iyo antihypertensive.
facooda Ruush waa dawo "Vero Amlodipine" macmalay by "Veropharm" OJSC, oo macnihiisu yahay "Amlodipine-Biocom" warshad "Biocom" CJSC.
medicament The "Amlodipine-Teva" jirta laba siyaalood: 0.005 iyo 0.010, labada qaadashada bandhigay kiniinada cadcad isagoo qaab biconvex wareegsan, calaamadsan "AB 5" ama "AB 10". Available shirkadda dawooyinka ee Hungarian "TEVA Prayvet Co. Co., Ltd. '.
Drug "Amlodipine Sandoz" soo saaray shirkadda Slovenia "Sandoz" oo ah qaab guri, unugyada kiniin wareega isagoo khatarta iyo chamfer.
Reviews
Bukaan badan sida qalab sababta oo ah waxtarka iyo qiimaha la awoodi karo. About daawo 'Stamlo "dib u eegista waxaa la maqli karo dabeecadda wanaagsan iyo wax xunba. Mid ka mid ah kaniiniyada bukaanka caawin yareeyo cadaadiska dhiigga ee sareeya, dadka kale ee aan awoodin in ay daaweyso hypertension.
Intaa waxaa dheer, daroogada ka cadhaysiinina karaan daal, wareer, daal, isbeddelo ah niyadda, hurdo, iyo lallabo. Xaaladdan oo kale, by qaadashada kaniiniga waa in la tuuraa.
Similar articles
Trending Now