Caafimaadka, Diyaarinta
"Glibenclamide": tilmaamaha loo isticmaalo, foomka la sii daayo, sawir, analogs
Waa maxay daawo "Glibenclamide"? Tilmaamaha loogu isticmaalo, foomka la sii daayo, analogues iyo tilmaamo maamulka daroogada waxaa hoos ku qoran.
Curiska, baakadaha, wakiilada foomka sii daayo
In waxa foomka la sameeyo daawo "Glibenclamide"? Guide ayaa sheegay in qalab la soo saaray qaab kiniin oo waxaa la geeyaa weel caag (dulmar ah cell) iyo sanduuqa laga sameeyay baakado, siday u kala horreeyaan.
Halabuurka The daroogada hoos tixgelin ka mid ah Glibenclamide 5 mg iyo maaddooyinka kaabayaal sida istaarijka baradho, laktosmonohydrat lactose, milmahayn magnesium, sodium croscarmellose, indigo Carmine E 132 Kolloidol Silicon dioxide 25, iyo povidone.
tallaabo Drug
Waa maxay daawada "Glibenclamide"? Tilmaamaha Isticmaalka sheegayaa in taasi ka dhigan tahay soo bandhigista saamayn hypoglycemic in dadka caafimaadka iyo bukaanka qaba diabetes nooca II.
Saamayntii daroogada this sabab u ah awoodda ay leedahay in la kordhiyo dheecaan insulin unugyada beta ganaca sabab u kicinta. Sida laga soo xigtay khubaro ah, saamayn this daroogada la wanaajiyey sarkhaansan yihiin sonkorta.
Ogeed qoreysa dejinta afka
Waa maxay astaamaha mid caan ku ah daroogada pharmacokinetic "Glibenclamide"? Tilmaamaha loogu isticmaalo waxa uu sheegayaa in ka dib markii kacmaha afka ah kiniin oo ah walaxda firfircoon si degdeg ah oo ku dhowaad si buuxda u nuugo ka soo mareenka dheefshiidka.
cuntada oo wadajira u keenaysaa in hoos u fiirsashada Glibenclamide ee plasma (la calool madhan la barbar dhigo). xidhiidhka ka mid qayb la albumin ka badan 98%.
Glibenclamide beerka bukaanka ah, waxaa beddelay ee metabolites soo socda: 3-CIS-hydroxy-Glibenclamide iyo 4-trans-hydroxy-glyburide. Waxay yihiin wax soo saarka ilaa xad isku by kelyaha iyo, wada jir ah ula saxarada ah.
The reebay celceliska bar-nolosha ee daroogada waa 2-3.5 saacadood. In dadka la beerka oo yaraada, tiradaasi waa weyn u dhimay.
Tilmaamayaasha ay u isticmaalaan daroogada
Xaaladaha qaarkood, a kiniinka bukaanka "Glibenclamide" waxa lagu meelaynayaa karaa? Taas macnaheedu waxa weeye talinaynaa qaadashada bukaanka qaba diabetes nooca II, marka ma jiro wax fursad ay ku buuxin hyperglycemia cunto adag iyo dhaqdhaqaaqa jirka, ama miisaanka oo yaraada.
Oo mamnuucday isticmaalka
Ma jiraan wax sababo in "Glibenclamide" daroogada? Tilmaamaha Isticmaalka dhigayaa in xarunta this waa in aan lagu maamulo in bukaanka qaba:
- gubasho ballaaran;
- Diidmo qayb firfircoon, oo lagu durayo ah thiazide ama sulfonamides;
- ketoacidosis;
- kooma macaanka iyo dalalka prekomatosnoe;
- horumarinta hypoglycemia,
- qalliinka iyo dhaawacyada kale;
- gastroparesis oo xirma xiidmaha;
- uurka;
- macaanka nooca ugu horeysay,
- naas-nuujinta.
Medicament "Glibenclamide": tilmaamaha loo isticmaalo
Waxaa loo tixgeliyaa daroogada waa in la maamulo kaliya dhakhtar khibrad leh. daroogada waa in had iyo jeer la weheliso cunto adag. Kaliya kiiskan waxa ay noqon doontaa wax ku ool ah. ay qiyaasta ku xiran tahay natiijada bukaan imtixaanka (heerarka sonkorta dhiigga, tilmaamayaasha ka soo jeeda kaadida, iwm).
Sidaas daraaddeed sida loo qaato daawada "Glibenclamide"? Therapy in ka dhigan tahay bilaw qaadasho yar. Tani waa run gaar ahaan dadka u janjeera in ay hypoglycemia iyo miisaanka jirka ka yar 50 kg.
Sida caadiga ah, marka ugu horeeysa ee reer medicament waa 0,5-1 kaniini maalintii. Taasi waxay u dhigantaa 2.5-5 mg firfircoon. Marka tirada tallaabo daroogada hawlqabad la'aan ku qeexan si tartiib tartiib kordhin karaa ilaa saddex kiniin maalin kasta, oo u dhiganta 15 mg ah ee firfircoon. Tani waa in la sameeyaa dura dhowr maalmood ilaa hal toddobaad, ilaa iyo natiijada la doonayo waxaa lagu gaarayaa.
Sida loo wareejiyo bukaanka si daroogada kale ee daawada "Glibenclamide"? Isticmaalka daawada kiiskan Waa in la fuliyo si taxadar leh u daran. First, bukaanka waxaa qoray loox 0.5 saacadood, ka dibna si tartiib ah u kordhiso qaadashada si uu waxtar wayn.
bukaanada waayeelka ah iyo u jilcay ama dadka qaba nafaqo-xumo iyo beerka ama kelyaha taageerooyinka shaqo oo yaraada ama qiyaasta hore ee daawada la doonayo si loo yareeyo suurtagalnimada of horumarinta hypoglycemia. Sidoo kale go'aan ku saabsan qiyaasta saxda ah ee daawada la hoos miisaanka jidhka ama marka laga beddelo hab dhaqanka nolosha waa in.
hab loogu talagalay la helo kiniini hypoglycemic
Sida loo isticmaalo daroogada "Glibenclamide"? Tilmaamaha loogu isticmaalo (photo of daroogada la soo bandhigay in this article) sheegaysaa in viewed kiniinka waa in la qaato cuntada ka hor la galaas oo biyo ah sifeeyo oo aan xanjo.
At qiyaasta maalin kasta ee 2 kiniin, waxaa lagu talinayaa in medicament ee 2 qiyaasood oo kala qaybsan (aroor iyo galabba) in cabirku yahay 2 qaybin: 1.
Waxaa aad u muhiima in la isticmaalo dawadan waqti isku mid ah. Kantaroolka ee samaynta kiniin dhaweynta Reebay wada qaatay la socda.
Muddada daaweynta wakiilka taasi ku xiran tahay cudurka. Intii ay daaweynta ayaa loo baahan yahay si ay u fuliyaan la socodka joogtada ah ee gobolka bukaan-socodka walxaha dhaafsiga.
waxyeellooyin
medicament analogs The "Glibenclamide" kuwaas oo hoos ku qoran, waxay keeni kartaa horumarinta dareen diidmo oo aan la rabin saameysey, hormoonada jidhka, nidaamyada durugsan iyo dheefshiidka neerfayaasha iyo hematopoietic. Marka tan la eego, bukaanka waxaa laga yaabaa muujin calaamado loo kasin sida lallabo, hypoglycemia darraanta kala duwan, cillad cagaarshowga, shuban, madax xanuun, cholestasis, daciifnimo, dawakhsanaan iyo daal.
Sidoo kale waa in la ogaadaa in qaadashada ee qalabka meesha kama saarayso muuqaalka kore ee falcelin maqaar iyo xasaasiyad sida photosensitivity, cuncun, finan maqaarka ah iyo calaamado kale xun.
Xaaladaha xad dhaafka wakiilada hypoglycemic
Waa maxay calaamadaha yimaadda marka sare qiyaasood oo daawo "Glibenclamide"? dalalka Buugga in badinta, bukaanka waxaa laga yaabaa in la horumariyo hypoglycemia, waxaana suurto gal Ulasocto daciifnimo, dareen gaajo, madax-xanuun, walaaca, dhidid xad-dhaaf ah, dawakhaad, gariirka muruqa, uurkuna waa, barar ka mid ah xanuunada maskaxda, aragtida iyo hadalka.
Daaweynta xaaladaha sida u baahan yahay gelitaanka cunto glucose-digestible deg-deg ah. Tusaale ahaan, casiirka furutada, sonkorta, sharoobada hadhuudh, shaah kulul macaan ama malab.
Xaaladaha sii daran, bukaanka waxaa maamula xal glucose 50%, "dextrose" "Glucagon" ama "Diazoxide". Waxa kale oo ay u baahan tahay gacanta gaarka ah ee glycemia, kariyaatiniin, nitrogen HOL, electrolytes iyo pH go'aaminta.
Dhexgalka siyaabo kale oo caafimaad
isku dhafan ee daroogada loo arkaa daawooyinka anti-systemic, tetracycline'nada, fluoroquinolones, chloramphenicol, MAO, iyo ACE, H2-blockers, "clofibrate" beta-blockers, probenecid, bezafibrate, "paracetamol", steroids dhiska, ethionamide, allopurinol, pentoxifylline, cyclophosphamide "reserpine", insulin iyo sulfonamides waa inay awoodaan inay potentiate hypoglycemia.
codsiga waafaqsan daawada la phenothiazines, thyroid iyo glucocorticoid hormoonnada, barbiturates, estrogens, diazoxide, progestins, glucagons, lithium cusbada, Adrenomimeticalkie ka dhigan tahay saluretikami acid nicotinic iyo taagayo wiiqi karo saamayn hypoglycemic.
daawooyinka noocan oo kale ah waxaa loo acidified kaadida (oo ay ku jiraan chloride ammonium, chloride calcium, ascorbic acid), kobcin karaan tallaabo ee medicament u tixgeliyo.
Isticmaalka "Glibenclamide" with "rifamycins" dedejisaa inactivation iyo in la yareeyo wax ku oolnimada hore.
macluumaad gaar ah
Wakiilka Hypoglycemic waa in la tixgeliyaa si taxadir leh bukaanada qaba cillad kelyaha iyo beerka, iyo sidoo kale cudur thyroid iyo qanjidhada adrenal, xaaladaha xummada iyo Khamriga chronic.
Si ay u fuliyaan daaweynta caadiga ah u baahan tahay la socodka joogtada ah ee heerka sonkorta dhiigga ee qofka bukaanka ah, iyo sidoo kale ay Digo.
Haddii qaadashada daawada bukaan-socodka uu yeesho hypoglycemia, sonkorta magacaabay gudaha (in kiiska haddii qofka miyir qabo). Haddii miyir, glucose waxaa intravenously maamulo, iyo glucagons - subcutant, intramuscularly ama faleebo. Ka dib markii bukaanka soo tooso, uu si deg deg ah ku siin doonaa cuntada, hodan ku carbohydrates, si looga fogaado ku xoogeystay of hypoglycemia.
Qiimaha iyo analogues (micne ah) hab
Select analogs daroogada this waa in ay ahaataa oo keliya xirfad iyo khibrad. Waayo, dhakhaatiirta sida daroogada waxaa ka mid ah kuwan soo socda: "Manin", "Manin", "Maniglid", "Betanaz" iyo "Antibet".
Sidoo kale waa in la ogaadaa in farmasiyada inta badan iska iibiso micne ah qalab this. The iyaga isticmaalka ugu badan, "Glidanil", "Glibeks", "Glibamid", "Gilemal", "Glibomet", "Glibenclamide". qiyaasta lacagta waxaa la doortay si gaar ah.
Sida qiimo "Glibenclamide" daroogada, waxa kala duwan ee kala duwan 280-360 rubles.
Reviews of daawo
Haddaba aad u ogaato in uu yahay daroogada "Glibenclamide". Tilmaamaha loogu isticmaalo, iyo qaab analogues oo ka mid ah hab kor lagu sharaxay.
Waxay dhihi ku saabsan dadka isticmaala daroogada this? Sida caadiga ah, dhamaan fariimaha ku saabsan waxaa hoos u dhigay dooda mid ah kuwii ama daawada kale daweynta in lagula talinayaa dadka qaba sonkorowga.
Macaamiisha ayaa sheegaya in inta badan "Glibenclamide" loo isticmaalo sida monotherapy ah. Inkastoo ay jiraan kuwa bukaanka waxaa qoray daroogada isku dhafan oo daroogo kale hypoglycemic.
Sida laga soo xigtay dhakhtarrada, magacaabidda daroogada hoos tixgelin baahan tahay in hab shakhsi ah. Xaaladdan oo kale, oo khabiir ku ah waa in ay yaqaanaan oo dhan natiijada falanqayn, iyo cilmiga kale. Qaado bukaanka "Glibenclamide" ee u bannaan waa mid aad u khatar u ah caafimaadka iyo nolosha.
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