Caafimaadka, Diyaargarow
"Fluanksol": Buug gacmeedka, faallooyinka dhakhtarka. Dhibaatooyinka kale ee "Fluanxol", oo ah daawooyinka daroogada
Waa maxay daawada "Flyuanksol"? Tilmaamaha loogu isticmaalo daroogada, waxyaabaha ay, waxyeelo, foomka sii daayo iyo guryaha pharmacological waxa lagu sharaxay si faahfaahsan in this article. ka waxaad ku baran doontaa waxa sababo iyo tilmaamo ayaa sheegay daroogada, qiime intee le'eg, waxa dhici doona hadii aad iska badisid ah, iyo wixii la mid ah. D.
Halabuurka The daroogada iyo foomamka sii daayo ay
Waa maxay walaxda firfircoon ku jira daawada "Flyuanksol"? tilmaamaha loo isticmaalo ee edbinta medicament dhigayaa in sida qayb firfircoon u soo fiiqan hydrochloride flupenthixol.
Sida in foomka of sii daayo, laakiin maanta waa hab a waxaa laga heli karaa oo keliya ee dhibcood, kiniin iyo xal, ku salaysan saliid-, loogu talagalay maamulka muruqyada dhexdooda. daroogada koowaad waxaa suuq in galaas zatemennom 10 ml, labaad - in kartoonka ah 100 ama 50 iyo saddexaad - in ampoules of 10 xabbadood.
Guryaha Guud ee daroogada
Waa maxay sababta daawada "Flyuanksol"? Kurtumm ku saabsan daroogada this hoos lagu soo bandhigay. Kiniiniyada iyo duro waa koox ka mid ah nooca daawooyinka. Waxay hantidaan anxiolytic, niyad jabka iyo saamayn ku dejinaysaa. ra'yi-celin wanaagsan oo ku saabsan daroogada this ku jira macluumaad in ay si fiican u shidaa gobolka dareenka bukaan socodka iyo gacan ka geysaneysaa in la qabsashada bulshada.
Sifooyinka pharmacological daroogada
Maxay yihiin astaamaha daroogada pharmacological "Flyuanksol"? Tilmaamaha loogu isticmaalo daroogada soo jeedisay in this waa neuroleptic a, ka xanibeen receptors adrenergic iyo receptors dopamine ee maskaxda. Natiijada oo ah walaxda firfircoon waxaa lagu gaarayaa suuxin. Sida caadiga ah, taasi dhacdo in ka badan 8-maalin qiyaasta ah si joogto ah.
Maxaad bukaanjiifka oo ku saabsan daawooyinka "Flyuanksol"? Reviews bukaannada ku jira macluumaad badan oo xiiso leh. Xaaladaha intooda badan, waxay la soco in daroogada halkii si deg deg ah meesha calaamadaha waallida iyo niyad-jabka, iyo sidoo kale kordhinayaan in dib u soo celinta ee fikirka. Bukaan-socodka oo ahaa xanuunada bulshada, waa bulsho ah iyo la qabsado bulshada.
Features daawo
Sidee daroogada "Flyuanksol"? Reviews of dhakhaatiirta iyo xirfadlayaasha kale ay sheegayaan in feature a of daroogada this waa in, iyada oo ku xiran qiyaasta waxa ay talaabo u qaadi kartaa bukaan siyaabo kala duwan.
saamayn waallida dajiya teedu ka dib codsiga medicament ka dhigan in lacagta ah 3 mg maalintii. By habka, xoogga saameynta kordhisaa la qiyaasta.
Inta ay ilaa 25 mg maalintii daroogada ma saamayn ku dejinaysaa. Si kastaba ha ahaatee, waxaa la ogaadaa in at qiyaasood oo sare, waxay keeni kartaa saamayn ku dejinaysaa non-gaar ah.
In wakiilka loo qoondeeyey neuroleptic dose kala duwan oo uu leeyahay saamayn anxiolytic fahmayaan. Marka la isticmaalayo qaadasho yar (ilaa qiyaastii 3 mg maalintii), daroogada adeegaan hawsha a daawada niyad jabka caadiga ah.
Sayidka, daroogada "Flyuanksol" waa inay awoodaan inay yareeyaan calaamadaha ugu muhiimsan ee psychosis, oo ay ku jiraan dhibaatooyinkooda khayaano, dhalanteed iyo cudurka fikirka. Waxa uu ku disinhibitory (i.e. kaakicin iyo antiautisticheskim) iyo yaraynaysaa disorder niyadda a, taas oo ugu dambeyntii kor u hawlgelinta ee bukaanka qaba calaamadaha niyad, ay la qabsashada bulshada fududeeyaa iyo wanaajisaa sociability.
Badan oo ku saabsan qaab isku duro
Diyaarinta "Flyuanksol Depot" waa xal saliid ah loogu talagalay irbado saldhig muruqyada dhexdooda. In si kale loo dhigo, daroogada this lagu shubo qaab flupenthixol.
Marka la isticmaalayo xal this qaabab yaryar iyo kuwa dhexdhexaadka ah (ilaa 100 mg 14 maalmood oo kasta) bukaanka ma aha suuxin Ta'wiil. waxaa Inkasta oo uu weli sii kordhaya at qiyaasood sare.
Maxay khubarada yidhaahdo oo ku saabsan foomkan of daroogada ( "Flyuanksol Depot")? Reviews bixiyaan in xal noocan oo kale ah ayaa muddo dheer soo-gaadhista bukaanka, halkii kaniini oo daawo. Waxaa intaa dheer, waxaa isagii u mahad, waa ay fududahay si ay u fuliyaan daaweyn waallida dajiya joogto ah, taas oo aad muhiim u ah bukaanka oo aan fuliyaan qoro caafimaad.
Laga soo bilaabo kor ku xusan waxaa lagu soo gabagabeeyey karaa in daawada "Flyuanksol Depot" waa awoodaa si looga hortago soo noqoshada soo noqnoqda ee la xidhiidha kala go 'lama filaan ah therapy. duridda la fulin karo dura laba ama afar isbuuc.
Pharmacokinetics
kaniiniyada intee leeg ayaa nuugo "Flyuanksol"? Ka dib markii maamulka afka fiirsashada ugu badan ee element firfircoon waxaa lagu gaarayaa in oo ku saabsan 3-7 saacadood ee plasma. bioavailability ee daroogada waa 40%.
element daroogada firfircoon wax yar ka guskiisa ka celiyaha mandheerta. Sidoo kale waa in la ogaadaa in, in tiro yar, waxaa la muujiyey iyadoo caanaha hooyada. Waana mid ka, metabolites leeyihiin dhaqdhaqaaqa neuroleptic.
Sidee duray "Flyuanksol Depot"? Guide sheegayaa in ka dib markii duridda of CIS walax (Z) decanoate -flupentixol Oo Qaliin cholesterol (enzymatic). Tani qaab element firfircoon ee CIS (Z) -flupentixol iyo decanoic acid. fiirsashada ugu badan ee serum waxaa marka hore gaari by dhamaadka toddobaadka ugu horreeya ka dib markii la isku duro.
Marka la helo Alwaaxdii galay muddo taranta ay ku saabsan tahay 35 saacadood. Haddii ay jiraan waxa loo adeegsaday xal la isku duro, fiirsashada hoos u aheyn in serum ah (3 asbuuc ka dib).
Soo bandhigay medicament firfircoon ee foomka of metabolites dhex xiidmaha, iyo kelyaha.
Tilmaamayaasha isticmaalka wakiilada neuroleptic
Xaaladaha qaarkood, daroogada muujinaysaa "Flyuanksol"? Its tallaabo laga yaabaa kala duwan, iyada oo ku xiran qiyaasta.
Daawada waxaa lagu tilmaamay at qiyaasood oo ilaa 3 mg maalintii xaaladaha cudur ee soo socda:
- diiqad fudud iyo heerka dhexdhexaad ah, oo ay la socdaan daal, walaaca iyo la'aanta initiative;
- xanuunada maskaxda in mariyo la reactions asthenic;
- xanuunada ka waalan (chronic), oo ay la socdaan arxandarro, murugada iyo walwalka,
- iyo cudura ba'an xaaladeed walaaca, iyo sidoo kale gobolka walwalka shucuureed xad-dhaaf ah, uma baahna daawo kabuubiso ama saamaynta hypnotic (tusaale ahaan, haddii bukaanku xumeynayo dajiye).
Medicament "Flyuanksol", analogues kuwaas oo lagu soo bandhigi doonaa dhamaadka maqaalka, waxaa loo doortay at qaadashada of 3 mg maalintii oo dheeraad ah haddii ay jirto weecasho ka mid ah kuwan soo socda: xaaladaha waallida in waxaa weheliya dhibaatooyinkooda khayaano, dhalanteed, rabshooyin in fikirka, anergy, arxandarro iyo autism.
Sababo isticmaalka wakiilada neuroleptic
Xaaladaha qaarkood, waxaa laguma talinayo in la isticmaalo daroogada "Flyuanksol"? Tilmaamaha loogu isticmaalo waxaa ka mid ah liiska soo socda ee sababo:
- da'da carruurta (18 sano);
- depression habdhiska dhimirka;
- nuujinta,
- inta aad uurka leedahay,
- sarkhaan barbiturates (acute);
- burburto,
- sarkhaan analgesics opioid'ka ba'an;
- pheochromocytoma;
- sumowga ba'an khamriga,
- dalalka suuxsan,
- lafta xakamaynta dhuuxa;
- isbedel bahal dhiigga;
- diidmo in neuroleptics isagoo qaab-dhismeedka tioksantenoviy.
Sidoo kale waa in la ogaadaa in aan lagu talinayaa in la qoro daroogada ah ee qaadasho yar (ilaa 3 mg) ku jira xaalad ah fawdada ah ama excitations.
Drug "Flyuanksol": waxbarida (kiniin, dhibciyo)
Wixii lagu daaweyn jiray walaaca iyo niyad xanuunada dose hore ee medicament ee kiniiniyada waa in ay ahaataa 1 mg maalintii hal mar (fiican in aroortii), ama 500 mcg laba jeer maalintii. Haddii saamaynta ku daweynta maqan yahay, xaddiga daroogada ee toddobaadkii waa la kordhin karaa ilaa 2 mg. Sayidka qiyaasta maalin walba (2-3 mg) loo kala qaybiyey dhowr marxaladood. Haddii saamaynta maqan yahay marka la isticmaalayo daroogada ee qiyaasta maximal (i.e., 3 mg), ka dibna waa in la baabiiyo.
In daaweynta ee xaaladaha waallida cadadka daawada dhigay shaqsi kaliya. qiyaasta bilowga maalin kasta waa in ay ahaataa 3-15 mg 3 qaadasho kala qaybsan. Haddii la doonayo, mugga sheegay waa la kordhin karaa ilaa 20 ama 30 mg maalintii. qiyaasta ugu badan waa in aanay noqon in ka badan 40 mg.
Sida wakiilka daaweynta dayactirka wakiil waxaa maamula qadarkuu of 5-20 mg maalintii hal mar (subaxii).
Sida dhibicda "Flyuanksol", waa in ay la qaaday oo kaliya gudaha. Dhakhaatiirta caadi ahaan kuu qori daroogada ee foomkan oo keliya in haddii, waayo, wax kasta sabab, ma qaadan kartaa daawada afka (kiniin). qiyaasta taageero loogu talogalay bukaanka waa 4-40 mg maalintii.
Duray "Flyuanksol": waxbarida, dib u eegista bukaanka
Xalka saliid leh, waayo, irbado saldhig muruqyada dhexdooda waa in la maamulay oo qoto dheer galay Rubuca sare sare ee barida. Qiyaasta iyo bareeg u dhaxeeya daawaynta waa in kaliya la rakibay si gaar ah (madax bannaan oo saameyn ku daweyn).
dejinta waxaa inta badan loo isticmaalaa in lacagta ah ee 20-40 mg (ama 1-2 ml) 2 ama 4 toddobaad kasta. Waa in la ogaadaa in bukaanka qaar ka mid ah waxay u baahan yihiin waxaa laga yaabaa in qiyaasood oo waaweyn oo bareeg gaaban u dhexeeya irbado.
Haddii mugga loogu talagalay daawooyinka la isku duro (20 mg / ml) waa in ka badan 2 ama 3 ml 1 nidaamka, waxaa lagama maarmaan ah si ay u tagaan oo ku saabsan xal u fiirsashada sare.
Diyaarinta 100 mg / ml waa in lagu duraa in mugga a of 50-200 mg (ama 0.5-2 ml) 2-4 toddobaad kasta. In noqoshada ba'an ama sii daridda cudurka mararka qaarkood waxay u baahan tahay hal mar sal-dhigida ka dhigan in lacagta ilaa 400 mg dura 2 ama 1 toddobaad. Ka dib markii ay qabaan calaamadaha daran noqotay, waa in aad soo saaro hoos u si tartiib ah in qiyaasta in ay dayactir ah (20-200 mg 2-4 toddobaad kasta).
Haddii loo baahan yahay in ay ka soo foomka afka daroogada diyaarinta parenteral daryeel taageero ah u gudbin, waxaa lagu talinayaa in lagu saleeyo nidaamka soo socda:
- lacagta maalinlaha ah (in mg) oo ah daroogada ee kiniiniyada x 4 = qiyaasta hal (in mg) duro 14 maalmood oo kasta.
Sidoo kale waa in la ogaadaa in hal toddobaad gudahood ka dib markii maamulka daroogada waxaa lagula talinayaa inay sii wado qaadashada daroogada kiniinada, laakiin qiyaas hoose. Raac-up mugga iyo farqiga u dhaxeeya nidaamka aasaasay si waafaqsan saamayn ku daweyn.
qiyaasta ugu badan xal isku duro (hal-yada) ku saabsan tahay 400 mg. Sayidka farqiga u dhaxeeya irbado waa in toddobaadkii.
Sida laga soo xigtay jawaabaha dadka bukaanka ah, marka si habboon loo isticmaalo, diyaarinta iyo dhaqmayo talooyinka caafimaad, waxa uu leeyahay saamayn togan ku saabsan guud ahaan xaaladda dareen.
waxyeellooyin
Can saamayn xun ku daawada jirka "Flyuanksol"? Dhibaatooyinka ay keento ay joogaan in daroogada, iyadoo aan loo eegin qaabka. Halkan ay hadda yihiin.
- habdhiska: giperkinetiko-hypertensive syndrome (light extrapyramidal), daciifnimo, akathisia, daal, wareer, dhimaal psychomotor, tardive dyskinesia, reactions dystonic iyo neuroleptic syndrome malignant.
- Heart iyo dhiig weelashii: tachycardia, hypotension, orthostatic.
- nidaamka hematopoietic: granulocytopenia.
- xubnaha dareenka: qas hoyga.
- GI: caloosha oo, cholestatic cagaarshow, afka oo qalala, isbedel transient in baaritaano beerka.
- nidaamka hormoonada jidhka, miisaanka oo kordha, galactorrhea, dhidid, gynaecomastia, impotence, dysmenorrhea, rabitaanka cuntada oo kordhay, hoos u libido, dareenka gubashada ah.
- nidaamka Urinary: haynta kaadida.
- Xasaasiyad: dermatitis, photosensitivity, iyo finan maqaarka ah.
tilmaamaha gaarka ah ee isticmaalka
Daawo taxaddar qoray in bukaanada qaba xanuunada wadnaha, cudurada convulsive, neefta, glaucoma, cudurka Parkinson, boogaha caloosha iyo mindhicirrada 12-tiperstnoj, neefta, Khamriga, emphysema, haynta kaadida, beerka, iyo kelyaha Prostatic benign.
Haddii bukaanka ayaa hore u helay neuroleptics ama dejiyayaasha leh saamayn ku dejinaysaa, waxaa lagama maarmaan ah in la joojiyo iyaga habsami qaadashada.
Marka daaweyn muddada-dheer, gaar ahaan qaadashada sare talinayaa gacanta iyo qiimeeyo xaaladda bukaanka si loo saxo dose dayactirka.
In daaweynta isku mar of diabetes shaqo ah ayaa sheegay in samaynta u baahan tahay waxaa laga yaabaa in qadar sixida insulin.
In codsiga ah ee neuroleptics laga yaabaa in neuroleptic syndrome malignant. astaamaha ugu wayn waxaa weeye rigidity muruqa, hyperthermia, xaaladda maskaxeed doorsoon, iyo cillad of habdhiska ku autonomic. Marka calaamadaha sida u baahan joojiyo deg deg ah ee magacaabidda ah ee daroogada iyo daaweynta calaamadaha taageero.
Xaaladaha intooda badan, daawo "Flyuanksol" ma keeno suuxin. Laakiin, inkastoo taasi, waxaa lagama maarmaan ah inay tixgeliyaan saamaynta ay iman kara on awood u leh inay si ammaan ah u shaqeeyaan mishiinka, ama habab kale. sidoo kale waxaan jeclaan lahaa in la ogaado in inta lagu guda jiro therapy (gaar ahaan bilowga), bukaanada waa inay ka fogaadaan shaqada aadka u halista ah (si loo ogaado jawaabta si daroogada).
xaaladood oo badinta
Haddii dawada si fiican loo qaaday (mugga kordhay), waxaa laga yaabaa inuu dhaco badinta. Xaaladdan oo kale, muujinayaa sifooyinka soo socda: hypo- ama hyperthermia, hurdo, gariir, disorder extrapyramidal, shoog, hypotension iyo kooma.
Maxaa la sameeyaa in xaaladda noocan oo kale ah? Waxaa lagama maarmaan ah si ay u fuliyaan therapy taageero iyo astaamaha. Haddii daroogada la daama, baahida loo qabo in si deg deg ah ku dhaq soo baxay caloosha, iyo sidoo kale in ay qaataan sorbent ah. Intaa waxaa dheer, waa mid aad u muhiim ah si ay u taageeraan hawlaha weelashii, wadnaha iyo neefsashada. Waxaa laguma talinayo in la isticmaalo epinephrine sida laga yaabaa in ay u horseedi in la yareeyo cadaadiska dhiigga. calaamadaha extrapyramidal waxaa suurtagal ah in la joojiyo daawada "Biperiden" iyo qalal - "Diazepam".
Dhexgalka daroogooyinka kale
Marka la isticmaalayo hal-yada ee medicament ayaa sheegay in la maqalka waxaa laga yaabaa in saamayn ku dejinaysaa of barbiturates, ethanol, iyo wakiilada kale oo saamayn inhibitory on yimaada habdhiska dhimirka.
Diyaarinta "Flyuanksol" waxa aan la talinayaa in la isticmaalo in lala guanethidine iyo walax Drug leh saamayn la mid ah. Dhab ahaantii Tan waxa u sabab xaqiiqada ah in nooca daawooyinka laga yaabaa in lagu xad wiiqay saamaynta ay antihypertensive.
Iyada oo hal isticmaal medicament "Flyuanksol" waxay yarayn kartaa waxtarka of daroogada "levodopa" iyo wakiilada kale adrenergic.
Isla mar ahaantaana qaadashada daroogada la a "piperazine" iyo "MCP" si weyn u kordhiyaa halista ah ee cudurka extrapyramidal.
Sidoo kale waa in la ogaadaa in daroogada neuroleptic soo bandhigay sida xal la isku duro kiis kasta waa in aan loo qaso dareeraha kale.
Price iyo analogues daroogada
Waa imisa daroogada ah "Flyuanksol"? Its qiimaha waa mid qaali ah. Sidaas daraaddeed, 50 kiniin oo ah 1 mg oo idinka mid ah in ay bixiyaan oo ku saabsan 500 rubles Ruush. Haddii aad rabto in 100 kiniin 5 mg, ay laga iibsan karaa 1,200 rubles. Sida foomka lagu mudo oo daroogada, waana ka qaalisan. In ka badan 10 fijaan (20 mg / ml) farmashiistayaasha u baahan tahay oo ku saabsan 2300 rubles.
Maxaa dhacaya haddii bukaanka uu awoodi daawo si ay u iibsadaan "Flyuanksol"? analogues Its waxaa lagu gadaa ku dhowaad dhammaan silsilado farmashiyaha. ka mid ah kuwa soo socda:
- Xalka "Flyuanksol Depot". Waa daroogada si dhakhso ah oo awood badan. Si kastaba ha ahaatee, waa kiniinno badan ka qaalisan.
- "Klopiksol" daawo. In qiimaha waa mid aad u dhow in asalka ah. Waxaa shaki on sale in kiniiniga iyo leedahay sababo dhawr.
- macnihiisu yahay "Truksal". Lagu iibiyo kiniin. Faa'iidada ugu weyn ee ay guushu ku isticmaalkeeda ee carruurta 3-sano. Kharash yar ka sarreysa asalka ah.
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