Caafimaadka, Diyaarinta
"Felodip": tilmaamaha loo isticmaalo, dib u eegista. analogues daroogada
Kaas oo ku baaqay in daroogada "Felodip"? Tilmaamaha loogu isticmaalo daroogada lagu tilmaami doonaa si faahfaahsan ee maqaalka soo bandhigay. Sidoo kale soo baxay waxaa ka mid ah, waxaad ku baran doontaa waxa daroogada this lagu meeleeyo, waxa dhinaca saamaynta uu leeyahay, in ama aan sababo daroogada this, qiime intee le'eg, taas oo uu leeyahay analogues iyo si bixi.
Halabuurka The oo daroogada ah, nooc ka mid ah wax soo saarka iyo baakada
In waxa foomka laga heli karaa daawada farmashiyaha "Felodip"? on isticmaalka hage dawadan sheegayaa in la heli karo oo kaliya in qaab kiniin la tallaabo dheer. Waxaa intaa dheer, qaadasho kala duwan ee daroogada ayaa baqshad oo kala duwan:
- kiniinka jaallaha ah ee foomka of digir laga sameeyey, iyada oo aan ur wax muujinaysaa tirada 2.5. The element firfircoon felodipine daroogada sida u dhaqmo qadarkuu of 2.5 mg. Excipients daroogada waa laktosmonohydrat lactose, hypromellose, cellulose mikrokristallin, xabagta cas bir ah, povidone, titanium dioxide, gallate propyl, xabagta huruud bir ah, milmahayn magnesium, tones propylene, silica Kolloidol ammooniya, Rusheyn kartaa. In iibinta daroogada firfircoon galo khariidad 10 kiniin in waxaa la geeyaa kartoonada.
- Loox oo midabka casaan khafiif ah ee qaabka digir laga sameeyey, iyada oo aan ur wax muujinaysaa tirada 5. qayb firfircoon ee diyaarinta sida ay laftu felodipine qadarkuu of 5 mg. Excipients daroogada taag laktosmonohydrat lactose, hypromellose, cellulose mikrokristallin, xabagta cas bir ah, povidone, titanium dioxide, gallate propyl, xabagta huruud bir ah, milmahayn magnesium, tones propylene, silica Kolloidol ammooniya, Rusheyn kartaa. In iibinta daroogada firfircoon galo khariidad 10 kiniin, waxaa la geeyaa galay kartoonada.
- Kiniiniga guduudasho cadas brown qaabeeya aan ur kasta loo qoondeeyey tireedyada 10. element The firfircoon ee noocan oo kale ah falalka felodipine daroogada qadarkuu of 10 mg. Auxiliaries waa laktosmonohydrat lactose, hypromellose, cellulose mikrokristallin, xabagta cas bir ah, povidone, titanium dioxide, gallate propyl, xabagta huruud bir ah, milmahayn magnesium, tones propylene, silica Kolloidol ammooniya, Rusheyn kartaa. In iibinta daroogada firfircoon galo khariidad 10 kiniin. Finan kaalinta galay kartoonada.
The guryaha pharmacological daroogada
Waa maxay qalab caafimaad "Felodip"? Tilmaamaha isticmaalka daroogada ayaa sheegay in uu yahay xanibaha channel calcium la'ahay. daroogada viewed iska leh kooxda ee dihydropyridine.
daawo Tani waa inay awoodaan inay tijaabiso saamayn antianginal iyo antihypertensive. Intaa waxaa dheer, waxa ay yaraynaysaa cadaadiska (dhiig) by hoos iska caabin dhuumaha ugu sarreeya.
Waa maxay guryaha kale ee ay leeyihiin daawooyinka "Felodip"? Tilmaamaha isticmaalka diyaarinta ka mid ah macluumaadka uu leeyahay saamayn anti-ischaemic dose-ku-tiirsane ah. Daawada yaraynaysaa size Wadnaxanuun, iyo sidoo kale ka ilaaliya jidhka dhibaatooyin reperfusion.
Qalabkani waxa uu leeyahay ficil ahaan ma saamayn inotropic xun. Waxay leedahay saamayn yar oo ku saabsan nidaamka qaban ka.
The pharmacokinetics daroogada
Sidee dheer daroogada la nuugo, "Felodip"? Tilmaamaha loogu isticmaalo, warcelin taasi ka dhigan tahay in ay bixiyaan ka dib markii dose oo ah medicament galay walaxda firfircoon waxaa ku dhowaad si buuxda u nuugo ka soo mareenka dheefshiidka iyo u dhaqmo si degdeg ah. Thanks to foomka qiyaasta ay, in la sii daayo dib u of element firfircoon ay hubisaa in ay fiirsashada uniform ee dhiigga (maalin gudahood), iyo sidoo kale waxay keenaysaa in la kordhiyo wajiga nuugo.
Waxaan ma dhihi karo in bioavailability ee daroogada kuma xirna qiyaasta ku daweynta iyo qiyaastii waa 15%.
Qabanaya borotiinka plasma oo dheeraad ah si hufan waa qiyaastii 99%. medicament waxaa la sii daayay oo ay la socdaan caanaha naaska iyo guskiisa caqabad dhiig-maskaxda iyo celiyaha mandheerta. Iyada oo la isticmaalo daba dheeraaday oo ah walaxda firfircoon raasamaal ma dhacdaa.
Halkee daroogada la metabolized "Felodip"? Walaxda firfircoon ee wakiilka this waxaa metabolized beerka. In foomkan metabolites firfircoonayn.
The bar-nolosha ee daroogada ku saabsan tahay 25 saacadood. diyaarinta soo bandhigay sida metabolites (ku dhowaad 70%) in kaadida iyo saxarada (30%).
Tilmaamayaasha medicament
Xaaladaha qaarkood, bukaanka waxaa soo qoray daawo "Felodip" (5 mg) Tilmaamaha daawada waxaa ku jira liiska soo socda ee muujinaya in loo isticmaalo:
- hypertension,
- angina,
- arrhythmia;
- wadne xanuunka,
- xanuunada wareegga dhiigga,
- Raynaud ee syndrome.
sababo daroogada
In kiisaska waa mamnuuc in ay qaataan daawada "Felodip"? Reviews dhakhaatiir, iyo sidoo kale tilmaamaha la socda sheegayaan in daawada waa in aan la isticmaali hoos shuruudaha soo socda:
- Wadnaxanuun myocardial ba'an, iyo sidoo kale hal bil ka dib markii myocardial gudahood;
- angina deganayn,
- lama filaan ah cardiogenic;
- wadnaha oo shaqadiisa gaba, gaar ahaan decompensated;
- stenosis aortic (Caafimaad ahaan la taaban karo);
- uurka;
- hypotension (daran);
- in carruurta iyo dhallinyarada (ka yar 18 sano);
- inta lagu jiro nuujinta;
- dareenka sii kordhaya ee bukaanka in ay daroogada ama taagayo kale dihydropyridine.
Mid ka mid ah waa in aysan iloobin in qalab this si taxadir leh u daran qoray in bukaanka qaba la'aan, cagaarshowga iyo kelyaha.
qalab caafimaad "Felodip": tilmaamaha loo isticmaalo
Analogues qalab this la yar oo dheeraad ah soo bandhigi doonaa. Hadda waxaan doonayaa in aan kuu sheego sida daawada waa in si sax ah loo qaaday.
Marka hypertension dose ee dadka waaweyn iyo dadka waayeelka ah ayaa lagu wadaa si gaar ah. Sida caadiga ah, lacagta bilowga ah ee daroogada waa 5 mg maalintii hal mar. Inta lagu guda jiro doorashada ee bukaanka ku haboon qiyaasta lagu talinayaa in la isticmaalo kiniin ah ee 2.5 mg. Marka deg-deg ah u baahan yihiin in la kordhiyo qiyaasta daawada waxay noqon karaan. mugga Celceliska medicament ah si loogu daweeyo dayactirka 5-10 mg maalintii.
Waayo, bukaanada waayeelka ah ama dadka qaba beerka si daciif ah in daaweynta daroogada hore waxaa maamula qadarkuu of 2.5 mg maalintii.
In daawada angina xasiloon "Felodip" shaqsi qoray. Sayidka ay dose hore (ee dadka waaweyn) waa 5 mg maalintii hal mar. Haddii loo baahdo, ee qiyaasta waa la kordhin karaa ilaa 10 mg maalintii. Lacagta ugu badan maalin walba ah ee daroogada waa 20 mg.
Kiniiniga "Felodip" waa la ogol yahay in ay qaataan isku dhafan oo celiyeyaasha ACE, beta-blockers iyo diuretics. Si kastaba ha ahaatee, waxaa la ogaadaa in halka ay saamayn hypotensive waa wanaajiyey. Haddaba sidaas daraaddeed waa inaad aad uga taxadirtaa sababtoo ah khatarta ah ee sii kordhaya ee hypotension.
In bukaanka qaba beerka si xun u daciif ah qiyaasta daawada waa in la dhimay.
Submitted by daroogada waa in kaliya la qaadi subaxdii ka hor quraacda. Xaaladdan oo kale, Oo looxa kiis kasta ma suurtowdo in crack, burburin ama u qaybi.
hab badinta
isticmaalka khaldan ee kaniiniga "Felodip" calaamadaha soo socda ee xad dhaafka ah ee bukaanka laga yaabaa inuu dhaco: bradycardia iyo hypotension (daran).
In case of dhacdo calaamadaha sida therapy astaamaha. Haddii hypotension (daran) bukaanada la siiyo meel siman oo kor lugaha. Marka la eego bradycardia, kaas oo kiiska atropine bukaanka intramuscularly maamula at qiyaasta ah 0.5-1 mg. Haddii loo baahdo, in la kordhiyo mugga of galiyey plasma waxaa lagu fuliyaa la chloride sodium, xal glucose ama dextran.
Marka tallaabooyinka iyo liidasho ay kor lagu sharaxay soo qoray daawo bukaanka qaba saamayn dega on receptors Alfa-adrenergic.
Dhibaatooyinka ay keento ka qaadashada daroogada
Karaa saameyn xun ku jidhka bini'aadamka qaadashada daawada "Felodip"? Analogues qalab this iyo diyaarinta laftiisa inta badan sababa madax xanuun, barrar wajiga, dawakhaad, wadno iyo daal. Si kastaba ha ahaatee, waxaa la ogaadaa in dareen diidmo oo kale waa karo. sida caadiga ah waxay u muuqdaan bilowga ah ee daaweynta, iyo sidoo kale iyadoo la kordhinayo qiyaasta of daroogada.
By jidka, iyadoo ku xiran cadadka daawada bukaanka laga yaabaa in muuqdaan iyo bararka durugsan helay. Sida laga soo xigtay khubaro, iyagu waa natiijada vasodilation precapillary.
In bukaanka qaba cirridka ama cudur cirrid in bukaanlayda qaadato daawada waxaa laga yaabaa in barar yar oo cirridka. Hawlgalkani waxa looga hortegi karaa, haddii aad u dhawrtaan nadaafadda afka dhamaystiran.
Mararka qaarkood waxaan ka fiirsaneysa inay qaadato daawada noqdo Jidka dhibaatooyinka soo socda:
- nidaamka wadnaha iyo, uurkuna waa, tachycardia, iyo barar durugsan.
- falcelin maqaar: photosensitivity, pruritus, urtikaria.
- Durugsan iyo bartamaha habdhiska: paresthesia, madax xanuun iyo wareer.
- Nidaamka muruqyada: arthralgia, myalgia.
- mareenka dheefshiidka: kelyaha ciridka, lalabo, korodhka in ensaymes beerka.
- Kale: daal, dareen diidmo oo diidmo, oo ay ku jiraan anjioedema.
Analogs, iyo kharashka daawada
Waa imisa daawo ina hor? Taasi waa arrin ka soo kiciyey by bukaanno badan daaweynta this qaliin lagu maamulo. Waa in la ogaadaa in maanta waa dawo ah waxa laga iibsan karaa qiimaha soo socda:
- Loox oo 2.5 mg (30 xabbadood) - 425 rubles Ruush,
- kiniiniyada in mugga a of 5 mg (30 xabbadood) - 556 rubles Ruush,
- kaniiniga in mugga a of 10 mg (30 xabbadood) - 831 rubles Ruush.
Maxaa bedeli karaa daawada "Felodip"? Analogs daroogada this waxaa laga helaa farmashiyaha shiidaa kasta. iyaga ka mid ah, waxaan doonayaa in aan ku muujiyo daawooyinka soo socda:. "Plendil," "Felodipine-NW", "Felodipine" iyo "faafiyo Felotenz"
ra'yi-celin wanaagsan ka yimi bukaanjiifka oo ku saabsan wax soo saarka, daawooyinka
Kurtumm ku saabsan "Felodip" gobolka diyaarinta in ay tahay aadka wax ku ool ah oo si fiican u dulqaadan by bukaanka, iyadoo aan loo eegin da'da iyo jinsiga. Intaas waxaa sii dheer, daroogada firfircoon waxaa laga yaabaa in xataa dadka qaba cudurka macaanka, cudurada kilyaha, neefta iyo cudurada kale ee sambabada obstructive la Raynaud ee syndrome, hyperlipidemia, turqo, iyo ka dib-tallaalidda sambabada.
khubaro badan ayaa farta ku xaqiiqada ah in daawada saameyn ah kuma laha profile la egyahay iyo sonkorta dhiigga fiirsashada.
dib u eegista negative
Ka mid ah dib u eegista xun in ka tago bukaan on daroogada this, waxaan la soco karo kuwa la xiriira qiimaha sare ee daroogada. Inkastoo farmashiistayaasha ku doodaya in ay qiimaha waa si buuxda u waafaqsan oolnimada iyo tayada.
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