Caafimaadka, Diyaarinta
Daawada "Pentas": tilmaamaha loo isticmaalo, analogs iyo dib u eegis
In dose oo ah daawo loo qoray "Pentas"? Tilmaamaha loogu isticmaalo, iyo dib u eegista ah ee daroogada ee hoos lagu sharxay. Sidoo kale article qalabka bixisaa macluumaad ku saabsan foomamka of sii daayo oo ka mid ah daroogada iyo hantida.
Halabuurka, qaabka medicament The
Waxa jira noocyo dhowr ah oo daawooyinka loo sii daayo tixgeliyo. Waxaan hadda u soo bandhigtid.
Diyaarinta "pentasil" - Kiniiniga (500 mg, 100 mg) tallaabo dheer. Inay u cad yihiin la-galyadeena grayish, iyo sidoo kale balastar badan oo bunni, qaabka saxda ah wareega, iyadoo Valium, qeebta iyo fariimihii labada dhinac.
element firfircoon ee daawooyinka tani waa mesalazine. Sidoo kale hab waa in qaab maaddooyinka povidone firfircoonayn, ethylcellulose, milmahayn magnesium, Rusheyn kartaa, iyo cellulose mikrokristallin.
In iibinta daroogada "Pentas" (kiniin), sawir ah kaas oo la soo bandhigay maqaal la gaarsiiyey baakad khariidad ku jira kartoon warqada.
Sidoo kale waa in la ogaadaa in medicament mawduuca laga iibsan karaa qaab dabada, dhagaxyada-daayo joogta ah iyo ganaax malawadka.
daawo Farmashiiste
Waa maxay daawo for "Pentas"? Tilmaamaha loogu isticmaalo dhigayaa in wakiilka la ficil anti-bararka iyo isticmaalo in lagu daaweeyo ulcerös kolit iyo cudurka Crohn.
guryaha anti-bararka ah ee daroogada ku muujiyey oo keliya isticmaalka degaanka. Tallaabadan waxaa keena Avv leukotrienes iyo prostaglandins, iyo sidoo kale Iscelin hawsha lipoxygenase (nuutrofilkaagu). Intaas waxaa sii dheer, qalabka waa awoodaa inuu faafiyo dheecaan ee immunoglobulin by limfosaytis iyo in la xakameeyo degranulation, iyo phagocytosis ee socdaalka nuutrofilkaagu.
wakiilada Gaar ahaan mindhicirka
medicament "pentasil" The (looxa), oo sideeda oo ka mid ah kaas oo la kor ku soo bandhigay, soo bandhigaa kaga hadlay waxqabadka bakteeriyada ka mid ah mid cocci iyo coli Escherichia. Sidoo kale, waxa uu leeyahay saamayn antioxidant ay sabab u tahay awooda inay xidhxidhaan walaxda firfircoon la xagjirka lacag la'aan (oxygen) iyo iyaga u baabbi'in.
isticmaalka habboon ee qalab this si weyn u yaraynaysaa halista labakaclaynta cudurka Crohn, oo ay ku jiraan dadka qaba ileitis (la duration cudur dheer).
Mabda'a hawlgalka goobaha caafimaadka
Sidee daroogada "Pentas"? Tilmaamaha on codsiga sheegayaa in saamaynta ku daweynta ee daroogada isla markiiba waa ka dib markii la mariyo xiriirka mesalazine la xabka xiidmaha.
Ka dib markii qaadashada kiniinka afka si degdeg ah loola jeedaa disintegrates in microgranules oo dhaqmaan sida foomamka gaar ah oo soo gaaray daayo walax firfircoon - mesalazine. Tani waxay bixisaa daroogada soo jiidashada u dhaxeysa 12- in malawadka dhamaan qiimaha pH ah.
hab Pharmacokinetics
Sidee nuugista ee daroogada "Pentas"? Tilmaamaha isticmaalka warar sheegaya in microgranules kaniiniyada burburay 12 gaadho malawadka ee 60 daqiiqo ee ugu horeysay.
Qiyaastii 30-50% ee qiyaasta ah nuugo ka mid ah daroogada ee xiidmaha yar. mesalazine Communication la borotiinada plasma waa 43% iyo acid N-acetylsalisylsyre-shan-aminosalicylic - 73-85%.
Mesalazine iyo taagayo ay ha dhex gelin BBB ah. guryaha daroogada Darka waxaa u muuqday oo kaliya marka la isticmaalayo qaadasho sare (1500 mg maalintii).
mesalazine Acetylation la kulmin in xuubka caloosha iyo beerka. walax Tan waxaa ka soo jeeda kaadida, caanaha naaska iyo saxarada.
Tilmaamayaasha loo isticmaalo daawooyinka
Xaaladaha qaarkood, daawooyinka laga yaabaa in lagu tilmaamay "Pentas" (kiniin)? khubaro Guest ay sheegayaan in daawada u qabata iyo sidoo kale marka:
- ulcerös kolit;
- cudurka Crohn.
Oo mamnuucday isticmaalka daroogada
Under waxa xaaladaha uma isticmaali karo qalab sida "Pentas"? Tilmaamaha (kiniin iyo noocyada kale ee daroogooyinka waxay leeyihiin sababo la mid ah) ayaa sheegay in laga reebay soo socda:
- diathesis hemorrhagic,
- cudurrada dhiig;
- nuujinta,
- Dheefshiidka boogaha mareenka;
- ee 2-5 toddobaad ee uurka ee ugu dambeeyey;
- la'aanta dehydrogenase glucose-6-phosphate,
- da'da laba,
- kelyaha ee daran;
- diidmo in Muqaadaraadka wakiilada;
- kaafi cagaarshowga daran.
daryeel gaar ah waa in la tixgeliyaa daroogada loo isticmaalo in bilaha ugu horreeya ee uurka, iyo sidoo kale beerka iyo kelyaha.
Medicament "Pentas": tilmaamaha loo isticmaalo
Xulashada qaab qiyaasta of daroogada waxay ku xiran tahay deegaamaynta habka ugu weyn ee pathologic, iyo sidoo kale dhererka lesions xiidmaha.
Dabada "pentasil" iyo ganaax la maamulo ee foomamka distal cudurka (proctosigmoiditis). Isla mar ahaantaana saddex shumac isticmaalo maalinta 500 mg.
Sida loo qoro dawooyinka afka "Pentas" (kiniin)? Tilmaamaha loogu isticmaalo dhigayaa in noocan ah daroogada waxaa lagula talinayaa oo kaliya noocyada badan ee cudurka. Waayo, ka hortagga labakaclaynta cudurka Crohn medicament ah waxaa laga codsadaa afar jeer maalintii (1 g mesalazine). Ku saabsan ka hortagga labakaclaynta ee UC, kiiskan, daroogada la qoray saddex jeer maalintii 500 mg.
At sii daridda ah dabcan cudur daawaynta socon waa for 8-12 toddobaad. Isla mar ahaantaana maalin kasta wuxuu qaadan lahaa 400-800 mg ah ee daawada (sadex jeer maalintii).
In cudur aad u daran waxaa laga yaabaa in la kordhiyo qiyaasta maalinlaha ah ee 3-4 g
Kiniiniga "pentasil" Waa in la doorbidayo in la qaado si toos ah cuntada ka dib, dareeraha ah qallocan biyaha caadiga ah.
Waxqabadka by-qof
Xaaladaha qaarkood, daroogada ee su'aasha waa dhibaatooyinka soo socda:
- stomatitis, gariirka ee addimada, afka oo qalala, wareer, lalabo, dabeecadeed niyadjab;
- rabitaanka cuntada oo luma, uurkuna waa dareen, laab, neefta oo ku qabata inta lagu guda jiro dhaqdhaqaaqa jirka, matag,
- hematuria, shuban syndrome, tachycardia, hepatitis, xabad xanuun,
- sii kordhaya ensaymes beerka, isbedbedelka cadaadiska dhiigga, ganaca, polyneuropathy;
- crystalluria, tinnitus, proteinuria (Digo protein), madax xanuun xanuunka dhanjafka,
- oliguria, leukopenia, anuria (kaadi la'aan), Torombositobiiniya, formation syndrome nephrotic ;
- hypoprothrombinemia, Agranulocytosis, eosinophilia, anemia.
Sidoo kale waa in la ogaadaa in qaadashada daroogada this in bukaanka laga dheehan karo: olisgospermiya, alopecia, photosensitivity, daciifnimo in addimada, lupus-sida syndrome, wax soo saarka hoos u dheecaan lachrymal, mumps.
Iska badinta daroogada
heshiisyo badinta la tahay in ay gutaan hurdo sii kordhaya, lallabo, gastralgia, matag iyo tabar jidhka oo dhan. Si aad u baabi'iyo calaamadaha waxay u baahan lavage degdeg gastric iyo sidoo kale magacaabidda caloosha jilciya daawooyinka iyo therapy posindromnoy.
isdhexgalka daroogada
medicament "pentasil" wuxu si aad u yarayso heerka of nuugista cyanocobalamin. Mesalazine sidoo kale waxay kordhisaa tayada wakiilada uricosuric (oo ay ku jiraan blockers of dheecaan embriyaha).
Sidoo kale waa in Waxaan la soco in daroogada kordhay firfircoon ulzerogennosti glucocorticosteroids yaraynaysaa saamaynta rifampicin iyo kor u sumoobo ee methotrexate fulyo saamayn hypoglycemic on taagayo sulfonylurea, spironolactone, furosemide iyo sulfonamides.
macluumaad gaar ah
At gelitaanka ee dhoos keli ah mesalazine waxaa lagu talinayaa in ay qaataan oo ay la socdaan waxyaabaha soo socda ama mustaqbalka dhow. Haddii waxa la la'yahay ah qaadasho yar, waa inaad isla markiiba la tasho dhakhtarkaaga. Waxaa reebban in ay joojiyaan daaweynta on iyaga u gaar ah.
Mararka qaarkood asalka ah wakiilada warbixinta bukaanka arkay Xumaan kaadida iyo contact lenses in cado huruud ah-orange.
In daaweynta mesalazine u baahan yahay kormeer caafimaad joogta ah oo hawsha nidaamka kelyaha ee bukaan-socodka ah. Sidoo kale, falanqaynta kaadida iyo dhiiga qofka bukaanka ah waa in si joogto ah (koorsada of therapy oo dhan, iyo sidoo kale ka dib markii ay dhamaystirka).
itimaalka ee dhacdo of dhibaato in bukaanlayda qaadato daawada this bateen kuwa "acetylators gaabiya".
Iyadoo horumarinta syndrome ba'an ee dulqaad la'aanta diyaarinta firfircoon qayb "Pentas" isla markiiba wuu rogay.
daawooyinka la mid ah oo dib u eegista macaamiisha
Ma la socotaa waxa la oran karo waa in lagu badalo daawada? On this waa in aad u sheegtaa dhakhtarka dhigata. Sida caadiga ah, in analogues qalab this ka mid ah daroogada ee soo socda: "Mesakol", "Salozinal" "Salofalk", "Mezavant", "Mesalazin" "Asacol".
Maxay yihiin dad leh oo ku saabsan qalab this, macaamiisha? Sida laga soo xigtay jawaabahooda, ayaa sheegay in medicament waa daroogada aadka wax ku ool ah in laga iibsan karaa farmashiyaha kasta. Bukaan-socodka waxay ku andacoodaan in mesalazine waa teedu aad u wanaagsan laftiisa ma aha oo kaliya in daaweyn laakiin sidoo kale ka hortagga cudurka Crohn iyo ulcerös kolit.
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