Caafimaadka, Diyaarinta
Daawada "Sporagal": tilmaamaha loo isticmaalo, analogs iyo dib u eegis
Sida loo qaato daawada "Sporagal"? Tilmaamo ku saabsan isticmaalka daroogada la sii tixgelin doonaa. Waxa kale oo aad baran doontaa in ay jiraan analogues ee diyaarinta this, qiime intee le'eg, waxaad isaga ku saabsan bukaanka, waxa ujeeddada waxaa maamula, iyo wixii la mid ah. D.
Form, halabuurka, antifungal baakooyinka daroogada
Diyaarinta "Sporagal" heli karaa foomka kaabsal. Its qayb weyn ee firfircoon yahay itraconazole. Sidoo kale wuxuu ka kooban yahay medicament polyetylen 20000 tones, sucrose, iyo acetate acrylate hydroxypropyl.
Marka la eego qolof ah, waxaa ka kooban yahay gelatin, titanium dioxide iyo indigotin.
In xirmo lagu iibiyo daawada "Sporagal"? Tilmaamaha la isticmaalayo qalab this waxaa gundhig in kartoon ah. Waxa kale oo ku jira kaabsal adag gelatin buluug ah (in finan), kaas oo ay leeyihiin ee dhagaxyada ah spherical midabka jaalaha ah.
Pharmacodynamics medicament
Sidee "Sporagal" kiniin? Sida laga soo xigtay tilmaamaha, daroogada waa derivative ah triazole. Waxa uu leeyahay dhaqdhaqaaqa sare ka dhanka ah fangaska.
daroogada wuxuu ka caawiyaa hakin Avv noolaha ee ergosterol, bixinta saamayn antifungal.
Khubarada ayaa sheegaya in itraconazole uu hakiyo koritaanka iyo taranka ee tirada badan ee noocyada of fangaska.
The pharmacokinetics wakiilka antifungal
Drug "Sporagal", taas oo analogues la sii cayimay doonaa, si dhakhso ah u nuugo dhex galaan wareegga dhiigga. heerka ugu sareeya ee itraconazole in aadanuhu ayaa lagu arkay 3 saacadood ka dib. Its bioavailability waa 55% (ugu badnaan waxaa lagu arkay at kaabsoosha soo dhaweynta si degdeg ah ka dib markii isticmaalka cuntooyinka baruurta iyo-calorie sare ah).
Itraconazole waxaa loo qaybiyey xubnaha iyo unugyada jirka ee kala duwan. Its content in lafaha, kelyaha, beerka, sambabada, murqaha lafaha, caloosha, beeryarada, iyo 3 jeer ka badan yihiin dhiigga.
Medicament metabolized beerka u sii daayo hannaanka ah taagayo. Si kastaba ha ahaatee, gidroksiitrakonazol kaliya ayaa saamayn antifungal dhawaaqaa.
Qiyaastii 34% oo ah walaxda firfircoon waa la sii daayay kaadida, iyo wax ku saabsan 54% iyada oo xiidmaha.
In dadka la function si daciif ah beerka iyo cudur kalyaha ah, iyo in bukaanka qaba bioavailability Baabi'id daroogada waa la dhimi karaa.
Tilmaamayaasha kaabsoosha
Maxaad u magacaabi "Sporagal"? Waxbarashada dhigayaa in daroogada waxaa loogu talagalay daawaynta cudurada boqoshaa, kuwaasi oo ay kaga xanaajiyeen by wareer dareen daroogada:
- candidiasis vulvovaginal;
- xanuunada ophthalmological iyo maqaar ka soo jeedo fangas (tus, keratitis fangas, fayada, versicolor pityriasis);
- candidiasis afka ;
- onychomycosis, kuwaasi oo ay kaga xanaajiyeen by dermatophytes ama gjærsopper;
- mycoses systemic oo ay ku jiraan cryptococcosis (dadka nidaamka difaaca jirka daciif ah inta lagu guda jiro habdhiska medicament cryptococcosis maamulo kaliya ay ka maqan yihiin saamaynta daaweynta wakiilada kale antifungal), cryptococcal meningitis, aspergillosis systemic iyo candidiasis;
- sporotrichosis, paracoccidioidomycosis, blastomycosis, histoplasmosis, iyo mycoses kale systemic dhif.
Sababo isticmaalka kaabsoosha
Maxay yihiin sababo ah in isticmaalka daroogada ah "Sporagal" (kiniin)? Waxbarashada dhigayaa in daroogada aan loo isticmaali in:
- Diidmo in qaybaha hoose iyo kuwa sare ee daroogada
- lala daawooyinka sida blockers "Eletriptan" inhibitors reductase HMG-CoA (tus, "atorvastatin", "Lovastatin" "dawo"), wada jir ergot, muhashada CYP3A4 (tusaale ahaan, "Cisapride", "bepridil," "pimozide" "Dofetilide", "Astemizole" "quinidine" "mizolastine"), "nisoldipine," "Midazolam", "triazolam".
Sidoo kale waa in la ogaadaa in isticmaalka daroogada this waa u siiyo dadka qaba cillad ventricular iyo wadnaha oo shaqadiisa gaba, gaar ahaan qof gabsiiya.
Drug "Sporagal": tilmaamaha loo isticmaalo
Sida laga soo xigtay tilmaamaha, daroogada waa in la qaato kaliya hadal. kaabsoosha waa in isla markiiba la wada baabbi'iyey hadhuudh ah (si loo hubiyo in nuugista wanaagsan) ka dib, in oo dhan, iyada oo aan xanjo.
qiyaasta daawada taasi ku xiran tahay nooca cudurka jira:
- Maqaar iyo nabar ophthalmologic (tus, versicolor pityriasis ama in fayada) - 200 mg maalintii hal mar for toddobaadkii.
- lesions Keratinized ee maqaarka (gacmaha iyo cagaha) - 200 mg laba jeer maalintii muddo wiig ah.
- candidiasis Vulvovaginal - 200 mg laba jeer maalintii muddo saddex maalmood ah.
- candidiasis Oral - 100 mg maalintii hal mar muddo laba toddobaad ah. In bukaanka qaba AIDS ama neutropenia, dose kordhay ilaa 200 mg maalintii hal mar.
- keratitis fangas - 200 mg maalintii hal mar muddo seddex isbuuc ah.
- Onychomycosis, kuwaasi oo ay sababa dermatophytes ama gjærsopper, waxaa lagu daaweeyaa by yahay koorsooyin soo noqnoqda. Mid ka mid ah therapy ku lug leedahay qaadashada laba kaabsoosha laba jeer maalintii muddo wiig ah. Wixii lagu daaweyn jiray lesions ciddiyaha faraha la fuliyay 2 kooxihii therapy this, oo cagihiisa on - 3 koorsooyinka. nasasho u dhexeeya labada waa in ay ahaadaan 3 toddobaad. Saamaynta la muujiyey marka la dhameystiro koorsada (with koritaanka taarikada ciddiyaha).
diyaarinta Qaxidda "Sporagal" oo ka mid ah ciddiyaha iyo maqaarka waxaa lagu fuliyaa muddo ka badan ka dhiigga. Marka tan la eego, saameynta ku daweyn fiicnayn dadka bukaanka ah waxaa lagu gaari kaliya seddex ka dib markii todobaad ka dib marka la dhameeyo therapy of cudurada iyo ku dhowaad 9 bilood kadib daaweynta onychomycosis.
Hababka Isticmaalka kaabsoosha for lesions systemic
Sida lesions systemic fuliyaan codsiga? "Sporagal" xil ee qaadashada soo socda:
- Candidiasis - 100-200 mg mar maalin kasta 5-30 toddobaad.
- Cryptococcosis aan meningitis - 200 mg maalintii 3-12 bilood. Iyada oo meningitis dose double.
- Aspergillosis - 200 mg maalintii 3-5 bilood.
- Histoplasmosis - 200 mg laba jeer maalintii muddo siddeed bilood ah.
- Chromomycosis - 100-200 mg maalintii muddo lix bilood ah.
- Sporotrichosis - 100 mg maalin kasta muddo saddex bilood ah.
- Paracoccidioidomycosis - 100 mg maalin kasta muddo lix bilood ah. Waayo, bukaan AIDS, qiyaasta lagu kordhin karaa.
- Blastomycosis - 100-200 mg maalintii laba jeer muddo lix bilood ah.
Dhibaatooyinka ay keento daawo
Ma jiraan waxyeellooyin in bukaanlayda qaadato daawada "Sporagal"? xirfadlayaasha Reviews sheegay falcelinta soo socda:
- neutropenia, Torombositobiiniya, leukopenia;
- caabuqyada neef-mareenka (sare);
- hypertriglyceridemia, hypokalemia, hypocalcemia;
- madax xanuun, paresthesia, neuropathy durugsan, hypoesthesia, dawakhaad,
- bukaanka serum, barar angioneurotic, anaphylactic iyo anaphylactoid cadaanyo;
- aragti cawlan, diplopia, maqal la'aanta, tinnitus, aragga indhaha oo isku darsamay;
- wadnaha oo shaqadiisa gaba, qof gaar gabsiiya;
- dyspnea, rhinitt, hogaga, barar sambabada,
- matag, dyspepsia, reactions hepatotoxic, calool xanuun, ganaca, lalabo, dysgeusia, calool, hepatitis, shuban, dibiro, sare u qaadis ku meel gaar ah transaminases beerka;
- xanuun ku jira laabatooyinka iyo muruqyada,
- finan, photosensitivity, vaskulitis leukocytoclastic, alopecia, necrolysis epidermal sun ah, pruritus, dermatitis exfoliative, finan, pustulosis exanthematous guud ba'an, multiforme erythema;
- dysmenorrhea, Xukun la'aanta kaadida, kacsi, pollakiuria;
- qandho, barar.
talooyin gaar ah
Waxyaabaha aad ogaanaysid bukaanka, ka hor inta aysan daroogada "Sporagal"? Responses sheegay in ay walax firfircoon waxay leedahay saamayn inotropic xun.
Inta aad qaadanaysid dawadan waxa dhici karta hawl gabsiiya wadnaha, iyo hepatotoxicity daran.
Marka hoos absorbability daroogada ashitada dilaacda.
Dadka isku mar codsanaya laabjeexa waa in la hayo iyaga iyo hababka diyaarinta bareeg tilmaamay of 2 saacadood inta u dhaxaysa.
Drug "Sporagal" laguma talinayo dadka bukaanka ah dadka waayeelka ah.
Haddii aad leedahay calaamadaha daawo durugsan qaadashada neuropathy si aad u joojiso.
Naas-nuujinta iyo uurka
Inta aad uurka leedahay, daawada lagu maamulo karaa oo kaliya in mycoses systemic, kuwaas oo khatar ku ah nolosha hooyada.
Sida naas-nuujinta, in muddo this, "Sporagal" waa la ogol yahay, laakiin kaliya ka yar tilmaamo adag.
Drug "Sporagal": analogs iyo qiimaha
Qalabka soo socda waa analogues ugu yaqaan daroogada hoos tixgelin, "Itrungar", "Sporaksol", "Orungal", "Eszol" iyo "Funit".
Waa imisa daroogada ah "Sporagal"? Qiimaha daawada this kala duwan 1100-1200 rubles.
Reviews of diyaarinta
Sida laga soo xigtay war celin kuwa qaatay daroogada, Waa in la ogaadaa waxa laga yaabaa in ay tahay arrin wax ku ool ah u muuqato in noocyada kala duwan ee cudurada fangas. la takooro karaa fariimo xun yihiin kuwa dhihi in qalab this leeyahay qiime sare. Si kastaba ha ahaatee, khubarada ku andacoodaan in qiimaha daroogada this waxaa si buuxda xaq ay oggolyahay daweynta.
Sida ee khasaaraha daroogada this, bukaannada inta badan farta ku muddooyinka dheer ee daaweynta.
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